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ethyl 2-[1-(2-ethoxypyridine-3-carbonyl)piperidin-2-yl]acetate
4-(2-methyl-1-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}propan-2-yl)morpholine
1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-3-(2-methylphenoxymethyl)piperidine
4-methyl-5-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
8-(2-hydroxybenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
2-methyl-4-[5-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)thiophen-2-yl]but-3-yn-2-ol
N-[2-(1H-indol-1-yl)ethyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
methyl 4-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]butanoate
N-[2-(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
2-(1H-1,2,3-benzotriazol-1-yl)-N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)acetamide
(1s,5s)-3,7-dimethyl-10-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3,7,10-triazatricyclo[3.3.3.01,5]undecane
3,4-dimethoxy-2-{[3-(2-phenylethyl)piperidin-1-yl]methyl}pyridine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}acetamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-5-methyl-1,2-oxazole-4-carboxamide
ethyl 1-(5-acetylthiophene-2-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
2,6-dimethyl-8-{[1-(thiophen-2-yl)ethyl]amino}octan-2-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}phenol
(2S)-1-(3-{[(3-methylthiophen-2-yl)methyl]amino}benzoyl)pyrrolidine-2-carboxamide
4-(3-methylpyridin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-2-carboxylate
4-methyl-2-[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]-1H-1,3-benzodiazole
N-(oxolan-2-ylmethyl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-[1-(furan-3-carbonyl)piperidin-4-yl]-N-phenylpropanamide
4-(1,3-thiazol-4-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}thiophene-3-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
(3S,4S)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(1H-indol-1-yl)ethan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-(3-methoxybenzenesulfonyl)pyrrolidine-2-carboxamide
1-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]azetidin-3-ol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methyl-1,2-oxazole-4-carboxamide
4-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrimidin-2-amine
7-(5-chloropyridin-2-yl)-4-(2-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-(2-hydroxyethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2,3,4-trimethoxy-N-(pyridin-4-ylmethyl)benzamide
3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-[(5-methylpyrazin-2-yl)methyl]-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
(3aR,6aR)-2-cyclopentyl-5-[(2,4-difluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{4-[5-(aminomethyl)-2-fluorophenyl]phenyl}methanol
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperazine-1-carboxamide
4-[1-(3,4-difluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-4-ol
2-(4-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}pyrrolidine-2-carboxamide
4-(6-cyclopropylpyrimidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{5-[1-(2-methoxypyridin-3-yl)-1H-imidazol-2-yl]thiophen-2-yl}-2-methylbut-3-yn-2-ol