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2-[(4aR,7aS)-4-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-cyclopropyl-1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(4aS,7aR)-1-[(4-hydroxyphenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-2-amine
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1-{1-[(3,5-dichloro-4-methylphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
5-[1-(cyclohex-1-en-1-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-2-(2-methoxyethyl)pyrimidine
4-{1-[4-(2-methylpropyl)benzoyl]piperidin-4-yl}-2-phenylpyrimidine
5-(2-chlorophenyl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]furan-2-carboxamide
N2-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-N4,N4,5-trimethylpyrimidine-2,4-diamine
4-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)piperidin-4-yl]pyridine
2-{2-[2-(piperidin-1-yl)ethoxy]phenyl}-1H-1,3-benzodiazole-5-carbonitrile
9-(1-cyclopentylpiperidine-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-{3-[4-(pyrimidin-2-yl)piperazin-1-yl]propyl}-1H-1,3-benzodiazole
5-{[(4aS,7aR)-4-(2-carboxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}furan-2-carboxylic acid
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
6-(methoxymethyl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]pyrimidin-4-amine
2-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(3-chlorophenyl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-4-carboxamide
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[1-cyclohexyl-5-(2,3,6-trimethylphenoxymethyl)-1H-1,2,4-triazol-3-yl]acetamide
4-(1H-pyrazol-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[1-(3-methylpyridin-2-yl)propan-2-yl]amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}ethan-1-one
(3R,5R)-5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]pyrrolidin-3-ol
N-methyl-5-({4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazol-1-yl}methyl)furan-2-carboxamide
N-[2-methyl-1-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
3-phenyl-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-[2-methyl-2-(morpholin-4-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-2,8-diazaspiro[4.5]decane
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(3-methoxyphenyl)methyl]piperidine
7-cyclohexyl-2-(1H-pyrazole-4-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 4-{[(2-cyclopropyl-1,3-benzoxazol-6-yl)formamido]methyl}benzoate
N-(6-fluoropyridin-3-yl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carboxamide
N-methyl-3-(4-methylpiperazine-1-carbonyl)-N-(naphthalen-1-ylmethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-7-hydroxy-5H,6H-benzo[h]quinoline-3-carbonitrile
methyl (2S,4S)-1-(cyclohexylmethyl)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}pyrrolidine-2-carboxylate
N-({5-[(2,6-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-(oxolane-2-carbonyl)-4-(thiophen-3-ylmethyl)-1,4-diazepane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-methyl-3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-indazole
7-[(3-methoxyphenyl)methyl]-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]propanamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-cyclopropylacetyl)piperidine-4-carboxamide
4-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1-methylpiperazine-2-carboxylic acid
2-(1-ethylpiperidin-4-yl)-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}acetamide
2-[(4aR,8aR)-7-(6-aminopyrimidin-4-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-N-(propan-2-yl)acetamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyridine-4-carboxamide
(1R,5S,6S)-6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane