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5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1-hydroxy-2-methylpropan-2-yl)-1H-pyrazole-4-carboxamide
2-(1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)pyridine
N-(3-methoxyphenyl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
5-{2-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]thiophene-2-carboxamide
1-(2-ethoxyethyl)-4-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperazine
3-(3-methoxyphenyl)-N-[3-(pyridin-2-yl)propyl]-1H-pyrazole-5-carboxamide
1-{4-[(4-methoxy-3-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazin-1-yl}ethan-1-one
2-(2,4-difluorophenoxy)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-(4-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
2-methyl-4-(3-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}phenyl)butan-2-ol
N-cyclooctyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
3-(2-ethylbutyl)-8-[1-(methoxymethyl)cyclobutanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{2-[2-(4-methoxyphenoxy)acetamido]ethyl}-N-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
4-methyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(cyclohex-1-en-1-yl)ethan-1-one
N-[(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)methyl]acetamide
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(4-fluorophenyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
1-[(5-methylfuran-2-yl)methyl]-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-5-methylpiperidin-2-one
3-(furan-2-yl)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)propan-1-one
(3S,4R)-1-(2-fluoro-6-hydroxybenzoyl)-4-methylpiperidine-3,4-diol
1-(4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
(4aS,8aR)-6-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
3-(1-cyclopentanecarbonylpiperidin-4-yl)-N-(3-methoxyphenyl)propanamide
8-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidine-3-carboxylic acid
7-fluoro-3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
1-{4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}imidazolidin-2-one
9-(cyclohex-3-ene-1-carbonyl)-2-(furan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})amino]-1-phenylpropan-1-ol
N-benzyl{[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]amino}sulfonamide
2-{4-[(4-methoxynaphthalen-1-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
{1-[(2-chloro-4-fluorophenyl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methylpyridine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
1-[(2-{[(1-methoxypropan-2-yl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
2-(4-{[methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]methyl}piperidin-1-yl)ethan-1-ol
N-methyl-4-(4-methylphenyl)-N-[(3-methylpyridin-4-yl)methyl]-5-(pyridin-3-yl)pyrimidin-2-amine
5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine
6-cyclopentyl-1-methyl-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}quinoline
1-(4-amino-5-methylpyrimidin-2-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[1-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide