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1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-3-yl)propan-1-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
(4aS,8aR)-6-[2-(methylsulfanyl)acetyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-butyl-N-methyl-3-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
3-{[1-(4-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methyl}benzamide
5-chloro-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-1,3-dimethyl-1H-pyrazole-4-sulfonamide
1-(3,5-difluorophenyl)-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
8-[(3-chloro-4-fluorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-amino-4-(1-benzofuran-2-yl)-6-cyclopropanecarbonyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1-ethyl-1H-1,2,4-triazole
5-(2-chloro-4,5-difluorobenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methoxybenzamide
2-(3-methoxyphenyl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]azetidine
3-[1-(2-chloro-6-fluorobenzoyl)piperidin-3-yl]benzoic acid
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methoxyethan-1-one
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N,N-bis(prop-2-en-1-yl)piperidine-4-carboxamide
(4aR,7aS)-1-methyl-4-(1-phenyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,3R)-N1-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
6-chloro-2-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]imidazo[1,2-a]pyridine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]benzamide
6-(aminomethyl)-2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-(propan-2-yl)-5-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyrimidin-2-amine
2-methoxy-5-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}phenol
(1S,5R)-3-[(6-ethoxypyridin-3-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(thiophene-3-carbonyl)piperidine-3-carboxylate
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
4-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-3,5-dimethylphenol
1-[2-methoxy-5-({[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-hydroxy-2-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-5-carboxamide
(3S,4R)-3-benzyl-1-(2,3-dimethylbenzoyl)-4-methylpiperidin-4-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
(1R,3S)-3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-N,N,2,2,3-pentamethylcyclopentane-1-carboxamide
1-{2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-ol
1-{4-[(2-hydroxy-3-methoxypropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
2-methoxy-3-(3,4,5-trimethoxyphenyl)pyridine
2-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}benzoic acid
2-[(4-chlorophenyl)methyl]-8-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
N,2,6-trimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]quinoline-3-carboxamide
2-amino-3-ethyl-N-(2-methoxyethyl)-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{3-[(3-chlorophenyl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
methyl 4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
methyl 4-(5-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate