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3-(1-ethyl-5-oxopyrrolidin-3-yl)-1-[4-(3-methoxyphenoxy)phenyl]urea
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-4-sulfamoylbenzamide
N-cyclopropyl-1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
4-methoxy-N-[(5-methyl-1H-imidazol-4-yl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-3-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-{[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
N-(1-phenyl-1H-pyrazol-5-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(4-hydroxypiperidin-1-yl)ethan-1-one
4-methyl-2-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-[4-({[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
1-(oxan-4-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine-3-carboxamide
4-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,4-oxazepane
(3S,7S,8aS)-3-(2-methylpropyl)-7-[(quinolin-5-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-1,4-oxazepan-6-ol
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-methyl-1H-pyrazole-5-carboxamide
1-(2H-1,3-benzodioxol-5-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-4-oxo-N-(thiophen-3-ylmethyl)-3,4-dihydroquinazoline-2-carboxamide
4-(1H-imidazol-1-yl)-N-[2-(pyridin-4-yl)ethyl]benzamide
N-[2-(3,4-dimethoxyphenyl)-2-hydroxyethyl]-2-ethylpyrimidine-5-carboxamide
2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
2-(4-fluorophenoxymethyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(3-hydroxybutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
7-(cyclopropylmethyl)-2-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-(1-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-2-phenylethyl)thiophene-2-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(3aS,6aS)-2-(oxan-4-yl)-5-[3-(pyridin-3-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
4-(3-phenylpropyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(1-phenylcyclohexyl)methyl]acetamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
[(3R,4S)-1-[(2-methoxy-3,5-dimethylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
6-ethyl-1-methyl-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-methylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
2-(2-methoxyethyl)-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}morpholine
(1R,2R,6S,7S)-4-(6-methyl-2-phenylpyrimidin-4-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(1R,7S)-3-(2-acetamidoethyl)-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-methyl-4-(4-methyl-1,4-diazepan-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-amine
1-{[2-(4-methoxy-3-methylphenoxy)phenyl]methyl}-4-methylpiperazine
N-(1-hydroxybutan-2-yl)-3-(propan-2-yl)-N-(thiophen-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[(2-methylphenyl)methyl]piperidine-1-carboxamide