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2-[(3,5-difluorophenyl)methyl]-8-[2-(dimethylamino)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
3-(1-{1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carbonyl}piperidin-4-yl)propanoic acid
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(naphthalen-1-yl)prop-2-ynamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
N-[3-(1H-indol-2-yl)phenyl]-1-(oxolane-3-carbonyl)piperidine-4-carboxamide
4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
4-[(3-hydroxy-4-methoxyphenyl)methyl]-1-methylpiperazine-2-carboxylic acid
3-(difluoromethoxy)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
N,4-dimethyl-5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
(2S)-2-{[6-(2-chlorophenyl)-7-(cyclopropylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-2-(1,4-dimethylpiperazin-2-yl)acetamide
3-[2-(2,3-dichloro-4-methylphenyl)-1H-imidazol-1-yl]propan-1-ol
5-cyclobutyl-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
2-methoxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[3-(methylsulfanyl)propyl]amine
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(methylsulfanyl)ethyl]amine
3-[2-(dimethylsulfamoyl)ethyl]-1-(3,4,5-trimethoxyphenyl)urea
{[5-(4-methoxyphenyl)furan-2-yl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
(2S,4R)-4-amino-N,N-diethyl-1-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}pyrrolidine-2-carboxamide
4-[6-(2-ethoxypyridin-3-yl)pyrazine-2-carbonyl]morpholine
3-{1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-1-ol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
1-(3-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}propyl)pyrrolidin-2-one
N-[(3S)-2-oxoazepan-3-yl]-4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)benzamide
1-(ethylcarbamoyl)-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
3-(3-fluorophenyl)-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
3-(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)-1-[2-(1H-imidazol-4-yl)ethyl]urea
2-acetyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
3-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-[3-(furan-2-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-3-[2-(2-methylpropanesulfonyl)ethyl]urea
6-[2-(2-chloro-6-fluorophenyl)acetyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl 3-(4-fluorobenzenesulfonamido)-5-{[(1-methylazepan-2-yl)formamido]methyl}benzoate
N-(3-methylbutyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-ethyl-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
[(3R,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyrazine-2-carbonyl)piperidine-4-carboxylic acid
methyl (2S)-1-(1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxylate
7-[2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(pyrazin-2-yl)piperazine-1-carboxamide
2-[4-(4-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazole
methyl 3-{[1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-(cyclopropanesulfonyl)-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
1-(3-chlorophenyl)-4-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]piperazin-2-one
(3R,5R)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide