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N-[(3R,4R)-3-hydroxy-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]pyridine-3-carboxamide
4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-methyl-1H-indol-1-yl)acetamide
4-{[(4-methyl-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}pyridine
methyl (1R,5S,6S)-6-{[4-(dimethylsulfamoyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
4-{4-ethyl-6-[4-(oxolane-2-carbonyl)piperazin-1-yl]pyrimidin-2-yl}morpholine
1-{1-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(3S,4R)-4-(hydroxymethyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-ol
2,2-diethyl-4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]morpholine
methyl 5-[2-(methylsulfanyl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
9-[2-(3-fluoro-4-methylphenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-cyclopentyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,3R)-2-amino-3-methoxy-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one
1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-3-ethoxypropan-1-one
2-{[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-1H-imidazole
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-{[5-(2-fluorophenyl)furan-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}pyridin-2-ol
6-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-ethyl-N-[(4-fluorophenyl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
(1S,5R)-3-benzyl-6-[(3,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[3-cyclopentyl-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-oxopyrrolidine-3-carboxamide
7-(pyridin-2-yl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(dimethylcarbamoyl)-5-{[(3-phenylpropyl)amino]methyl}phenyl]pyridine-2-carboxamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
(3S,4R)-1-[2-amino-4-(trifluoromethyl)pyrimidine-5-carbonyl]-4-methylpiperidine-3,4-diol
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
N-[(3R,5S)-1-(cyclopentylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
3-[(propan-2-yl)sulfamoyl]-5-(1H-1,2,3-triazol-1-yl)benzoic acid
N-butyl-N-(furan-2-ylmethyl)-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-2-(thiophen-2-yl)pyrimidine
6-(2-cyclopentyl-2-phenylacetyl)-N-[2-(1H-indol-3-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
6-[(diethylamino)methyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(1H-pyrazol-1-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide
2-methoxy-3-[3-(4H-1,2,4-triazol-4-yl)phenyl]quinoline
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethylamino)ethan-1-one
N6-cyclopropyl-N4-(isoquinolin-5-ylmethyl)-N4-methylpyrimidine-2,4,6-triamine
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-cyclopentylacetamide
3-[2-(3-phenylpropyl)morpholine-4-carbonyl]pyridin-2-ol
1-[2-(morpholin-4-yl)ethyl]-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
5-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-({1-[ethyl(methyl)sulfamoyl]pyrrolidin-3-yl}methyl)benzoic acid
2-cyclopropyl-1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-imidazole
3-cyclohexyl-N-[2-(ethanesulfonyl)ethyl]-1H-pyrazole-4-carboxamide
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine