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5-(2-chloro-4-fluorophenoxymethyl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[3-(hex-5-enamido)phenyl]-4-methylbenzamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}urea
2-[4-(4-chloro-2-fluorobenzoyl)-2-oxopiperazin-1-yl]benzonitrile
2-(4-fluorophenoxy)-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
5-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methoxy-4-methyl-1,3-thiazole
1-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-3-(2-methylphenyl)pyrrolidin-3-ol
N-methyl-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-methyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-(3-methyl-4-{[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
(3S,4S)-1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-(5-{1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
1-{3-[1-(dicyclopropylmethyl)-1H-imidazol-2-yl]phenyl}ethan-1-one
ethyl 1-(furan-3-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-[2-(2,6-dimethoxyphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-(furan-3-ylmethyl)-4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine
2-methoxy-6-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenol
(3R,4R)-4-cyclobutyl-3-methyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-3-ethyl-N,1-dimethyl-1H-pyrazole-5-carboxamide
N3-methyl-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-N3-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4S)-1-benzyl-4-[(1-benzylpiperidin-4-yl)amino]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
5-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-(2-chlorophenoxy)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,5-dimethyl-1H-indazole
4-(2-methyl-1H-imidazol-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)butanamide
2-(4-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)pyridine
5-(cyclohex-3-ene-1-carbonyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(1H-pyrazol-4-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
2-(cyclopropylmethyl)-9-(2,4,6-trimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]amino}methyl)-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
1-(diethylamino)-3-[2-methoxy-4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
1-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-2-carboxamide
N-[(1R)-1-carbamoylethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-(3-fluorophenoxy)-1-[2-(pyridin-4-yl)acetyl]piperidine-4-carboxylic acid
4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]sulfonyl}-N-methylbenzamide
3-(1H-indol-3-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
methyl 6-[(3-chlorophenyl)methyl]-2-(thiomorpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2-methylpropyl)-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(benzylsulfamoyl)[4-(furan-2-yl)butan-2-yl]amine
N-cyclopropyl-6-methyl-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
1-(2-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(1R,5S)-6-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-6-azabicyclo[3.2.1]octane
1-(4-methoxyphenyl)-2,2-dimethyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
6-ethyl-3-[2-(3-hydroxypiperidin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-cyclopentyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
4-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]-2,1,3-benzoxadiazole