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N-[3-(3-chlorophenyl)phenyl]-1-(furan-3-ylmethyl)piperidine-4-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methylthiophen-2-yl)methyl]benzamide
1-(2-methylpyridin-4-yl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-diazepane
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,5-dimethyl-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]acetic acid
(2R)-1-[(3S)-3-ethylmorpholin-4-yl]-2-hydroxy-2-phenylethan-1-one
(3S,4S)-1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-4-(dimethylamino)pyrrolidin-3-ol
N-(pentan-3-yl)-N-(2-phenylethyl)-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-(methylsulfanyl)propan-1-one
8-[3-(methylsulfanyl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-5-[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
3-[7-(cyclohexylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
N-(3,4-dimethylphenyl)-1-(2-methylfuran-3-carbonyl)piperidin-3-amine
2-({2-[4-carbamoyl-4-(piperidin-1-yl)piperidine-1-carbonyl]phenyl}amino)acetic acid
N-methyl-3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
N-(2-hydroxyethyl)-1-[(2-methoxyphenyl)methyl]-6-oxo-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-1,3-dicarboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanamide
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
1-{4-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
N-cyclopropyl-2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]acetamide
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-methoxy-3-methylphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
(3S,4R)-4-(hydroxymethyl)-1-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}piperidin-3-ol
5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}isoquinoline
2-{4-[7-methyl-4-(3-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
N-cyclopentyl-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-2-[2-(4H-1,2,4-triazol-4-yl)phenyl]acetamide
(4aS,7aR)-1-(2-methoxypyridine-3-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-methylprop-2-en-1-yl)propanamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
3-(1-methyl-1H-pyrrol-2-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-pyrazole-5-carboxamide
1-(4-fluoro-2-methylphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)pyridine-3-carbonitrile
4-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-4H-1,2,4-triazole
6-(pyrimidin-5-yl)-3,4-dihydroquinazolin-4-one
N-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
methyl (1R,5S,6R)-6-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
8-(2,5-dimethylfuran-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(azepane-1-sulfonyl)-5-bromobenzoic acid
4-[(5-methylthiophen-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-4-ethyl-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidine-3,4-diol
4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-2-(thiophen-2-yl)-1,3-thiazole
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-methyl-2-[5-(1-propylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-(3-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide