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({4-ethyl-5-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-chloro-2-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}phenol
(3S,4R)-1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-{3-[(3-methoxypiperidin-1-yl)sulfonyl]benzoyl}-4-methyl-1,2,3,6-tetrahydropyridine
1-(2,6-dimethylpyridin-4-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carboxamide
2-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1-methyl-1H-imidazole
{[5-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(1S,5R)-3-(6-amino-2-methylpyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,3s,6r,8S)-4-(quinoline-5-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
N-cyclopropyl-3-{1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}propanamide
1-[(4-methoxyphenyl)methyl]-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
1-[1-({1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-(4-{[2-(2-hydroxyethyl)morpholin-4-yl]methyl}phenoxy)acetic acid
(1H-1,3-benzodiazol-2-ylmethyl)(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amine
3-chloro-2-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-1H-indole
2-methyl-5-(4-{[(quinolin-2-yl)amino]methyl}piperidin-1-yl)-2,3-dihydropyridazin-3-one
4-(4-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-1-yl)-6-ethylpyrimidine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[7-(furan-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,5-dihydro-1H-pyrrole
[(3R,4R)-1-(6-cyclopropylpyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
7-(cyclopropylmethyl)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(1-ethylpyrrolidin-2-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
N-methyl-6-oxo-4-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-(dimethylamino)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(2-methylphenyl)acetamide
4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1-(propan-2-yl)pyrrolidin-2-one
N3-ethyl-N1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}pyrrolidine-1,3-dicarboxamide
2-[(4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethan-1-ol
methyl (2R,4S)-4-hydroxy-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidine-2-carboxylate
8-{[5-(hydroxymethyl)furan-2-yl]methyl}-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
{5-methyl-7-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-{2-hydroxy-3-[2-methoxy-4-({[2-(2-methoxyphenyl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
1-[(4-methoxyphenyl)methyl]-4-[3-(1-methylpiperidin-2-yl)propanoyl]piperazin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(adamantan-1-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]ethan-1-one
(1R,2S)-2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
(4aS,8aR)-6-[(4-fluoro-3-methoxyphenyl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
methyl(1,3-thiazol-2-ylmethyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-methylfuran-2-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-[2-(pyridin-3-yl)acetyl]-1,4-diazepan-2-one
2-{1-[(3,4-difluorophenyl)methyl]-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(3S,4R)-1-(cyclobutylmethyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
2-ethyl-9-[3-(2-fluorophenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
N-(3-phenylpropyl)-N-(propan-2-yl)-1H-pyrrole-2-carboxamide
(1R,9aR)-1-({[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
6-(2,3-dimethoxy-5-methylphenyl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide