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2,5-dimethyl-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
6-ethyl-2-methyl-4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]quinoline
5-methoxy-2-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]-1H-indole
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-(morpholin-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
1-(furan-2-yl)-2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethane-1,2-dione
5-(2-chlorophenyl)-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]furan-2-carboxamide
9-[(2,5-dichlorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methyl-1,3-thiazol-4-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
methyl({1-[1-(oxane-4-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-3-ylmethyl)amine
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-phenylpiperidine-1-carboxamide
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]-1-propylpyrrolidin-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1,5-trimethyl-1H-pyrazole-3-carboxamide
5-(1-benzyl-1H-pyrazol-4-yl)furan-2-carboxamide
N-[1-(1H-imidazol-2-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
14-{2-[2-(dimethylamino)ethoxy]phenyl}-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(2,3-dihydro-1H-inden-1-yl)-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propan-1-one
8-fluoro-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-2-carboxamide
[(4-{[1-(3-fluorobenzoyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(2-phenylethyl)amine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4,6-dimethylpyrimidin-2-amine
2-{2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
8-(2,5-dichlorophenyl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-{[6-(isoquinolin-5-yl)pyridazin-3-yl]amino}ethan-1-ol
4-{[(1R)-1-phenylethyl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
1-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]piperidine-4-carboxamide
methyl 4-({[(3R,5S)-1-[(4-chlorophenyl)methyl]-5-[(2-methoxyethyl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxypropyl)piperidine
1-ethyl-3-methyl-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrazine
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4-methyl-1,3-oxazole-5-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
2-(methoxymethyl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
4-[6-amino-5-cyano-4-(4-hydroxy-3-methoxyphenyl)pyridin-2-yl]benzoic acid
1-(4-methoxyphenyl)-2,2-dimethyl-4-(6-methylpyridine-2-carbonyl)piperazine
1-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-3-yl]pyrrolidin-2-one
4-({[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-ethoxyphenol
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,2-dimethyl-1-benzofuran-5-carboxamide
3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N-(pyridin-3-yl)propanamide
N-(adamantan-1-ylmethyl)-N-(2-hydroxyethyl)-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
3-{5-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-cyclopropyl-4-[methyl({[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl})amino]pyridine-2-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(2-methoxyethoxy)ethan-1-one
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-methylurea
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-methylthieno[2,3-d]pyrimidin-4-amine
3-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-(furan-2-ylmethyl)propanamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol