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4-methyl-4-(phenoxymethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
4-{4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[4-(1-benzylpiperidin-4-yl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[2-(2-fluorophenyl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
[2-ethoxy-5-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)phenyl]methanol
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1,1-dioxo-1λ6-thiolane-3-carboxamide
1-methyl-4-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(3aR,6aS)-2-methyl-5-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{2-methyl-4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}propan-1-one
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]acetamide
5-{3-cyclopropyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-hydroxyphenyl)-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
4-{2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}morpholine
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-N-methyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]piperidin-3-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(2-methyl-1H-indol-1-yl)propanamide
N-(2-hydroxyethyl)-1-(2-methoxyphenyl)-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
N-[(3S,4R)-1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
2-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
3-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]pyridine
2-(6-aminopyridin-3-yl)-2-[methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})amino]acetic acid
N-methyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-N-(2-phenylethyl)piperidin-3-amine
3-{2-[2-(furan-2-yl)azepan-1-yl]-2-oxoethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-(3-fluorophenyl)piperazin-2-one
methyl N-(2-oxo-2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}ethyl)carbamate
(2S,4R)-4-amino-N-methyl-1-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)pyrrolidine-2-carboxamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
1-[(4-fluorophenyl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(ethylamino)-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
5-fluoro-2-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-2-yl)-1H-1,3-benzodiazole
2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
7-cyclohexyl-2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-(2-{5-[2-(methylamino)pyridin-4-yl]-1,2,4-oxadiazol-3-yl}ethyl)pyrrolidin-2-one
2-(pyridin-4-ylmethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-chloro-5-acetamido-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-ethyl-8-{[2-(furan-2-yl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
propan-2-yl 4-chloro-3-(3-acetamidopropanamido)benzoate
N-[(2-chlorophenyl)methyl]-N-(propan-2-yl)quinoxaline-2-carboxamide
4-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl}benzoic acid
2-(3-chloro-4-hydroxyphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
5-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
3-[1-(2,6-dimethylpyridin-4-yl)piperidin-3-yl]-N,N-dimethylpropanamide
3-cyclohexyl-N-(2-hydroxy-3-phenoxypropyl)-1H-pyrazole-4-carboxamide
4-[1-(methoxymethyl)cyclobutanecarbonyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one