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1-butyl-3-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-1-(pyridin-4-ylmethyl)urea
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(pyridin-4-ylmethyl)propanamide
2-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine-3-carbonyl}pyridine
[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]diphenylmethanol
dimethyl[2-(2-{1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
1-(2,3-dihydro-1H-inden-2-yl)-4-[2-methyl-2-(morpholin-4-yl)propyl]-1,4-diazepane
2-{[1-(4-methoxyphenyl)piperidin-4-yl](methyl)amino}-N,N-dimethylpropanamide
2-methyl-N-(4-{methyl[3-(oxolan-2-yl)propyl]carbamoyl}phenyl)furan-3-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(methylsulfanyl)ethyl]pyrrolidin-2-one
1-methyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
3-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-5-carboxamide
2-(4-hydroxyphenyl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]propanamide
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-[2-(1H-imidazol-4-yl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
3-{5-[2-(3-methylphenyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}propanamide
2-[4-(2-methyl-2-phenylpropanoyl)-2-oxopiperazin-1-yl]benzonitrile
1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,2-bis(prop-2-en-1-yl)piperidine
(butan-2-yl)(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(pyridin-3-ylmethyl)amine
3-[(dimethylamino)methyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-ol
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-benzyl-4-[(4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,3-oxazol-2-yl)methyl]piperazine
2-butyl-8-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2,3-dichlorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[4-(piperidin-1-ylmethyl)benzoyl]-4-(pyridin-4-ylmethyl)piperazine
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
3-(3-{[benzyl(cyclobutylmethyl)carbamoyl]amino}phenyl)-N-methylpropanamide
(3S,4S)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}benzene-1,2-diol
3-[5-(oxolan-2-yl)-1H-1,2,4-triazol-3-yl]pyridine
N-[(2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]propanamide
(3R,7S,8aS)-3-(2-methylpropyl)-7-[(thiophen-2-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl 2-[(3-fluoro-4-methylphenyl)sulfamoyl]-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
7-[(3-methoxyphenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 4-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxylate
N-(4-{2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-oxoethoxy}phenyl)propanamide
4-(2,3-dihydro-1-benzofuran-7-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrrolidine-1-sulfonamide
[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
benzyl 1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxylate
9-(3,4-diethoxybenzoyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)-1-phenylpropan-1-ol
1-[(4-chlorophenyl)methyl]-5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(propan-2-yl)pyrimidine
14-(5-fluoro-2-methoxyphenyl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
1-(4-cyclohexyl-1,4-diazepan-1-yl)-2-(3-fluorophenoxy)ethan-1-one
(2R)-2-amino-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-phenylacetamide