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(3aR,6aR)-2-(prop-2-en-1-yl)-5-[4-(1H-pyrazol-1-yl)butanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[1-(cyclohexylmethyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
N-cyclopropyl-2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-({4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-1-yl}methyl)benzonitrile
N-[(1S,2R)-2-aminocyclobutyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
(2S,4R)-4-amino-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
N-[1-(4-methanesulfonylphenyl)ethyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]phenol
(3R,4S)-3,4-dimethyl-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-ol
1-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-4-phenylpiperazine
N,N-dimethyl-7-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
1-ethyl-5-(2-methoxyacetamido)-N-methyl-2-(pyridin-3-yl)-N-[1-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}methyl)pyridine-3-carboxylic acid
5-(2-chloro-4-fluorophenoxymethyl)-N-[3-(1H-indazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
2-amino-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
4-(1H-imidazol-1-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)benzamide
1-benzoyl-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidine
N-(5-ethyl-1,3,4-oxadiazol-2-yl)-2,2,6,6-tetramethylpiperidin-4-amine
1-{7-[(4-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-phenylethane-1,2-dione
2-methyl-N-{4-methyl-2-[4-(1H-1,2,4-triazol-1-yl)butanamido]phenyl}benzamide
N-cyclopentyl-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
1-[2-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-[(2-methoxypyrimidin-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N4,6-dimethylpyrimidine-2,4-diamine
2-(4-chlorophenyl)-4-(2-propoxyethyl)morpholine
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
(2S,4S)-N,N-diethyl-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
4-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]pyridine
N-({1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}methyl)acetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-(1H-indol-3-yl)-N-methylpropanamide
4-[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-oxo-N-phenylbutanamide
1-ethyl-3-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-3-carboxamide
2-butyl-N-[3-(4-methylpiperidine-1-carbonyl)phenyl]-2,5-dihydro-1H-pyrrole-1-carboxamide
ethyl 1-[1-(propan-2-yl)piperidine-4-amido]cyclobutane-1-carboxylate
8-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-2-(methylamino)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyridine-4-carboxamide
N-benzyl-3-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-(piperidin-1-yl)-N-[1-(pyrimidin-4-yl)ethyl]benzamide
1-(4-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
5-(3-methoxyphenoxymethyl)-N-[2-(6-methylpyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
8-(4-aminopyrimidin-2-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(3S)-3-ethyl-4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]morpholine
2-{4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-N-(pyrazin-2-yl)acetamide
3-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzoic acid
4'-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4,6-dimethyl-3-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1,2-dihydropyridin-2-one