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methyl 2-{3-oxo-1-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]piperazin-2-yl}acetate
1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-hydroxypiperidine-4-carboxylic acid
4-(2,4-dioxoimidazolidin-1-yl)-N-(2,2,2-trifluoroethyl)benzamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)-N-[2-(morpholin-4-yl)ethyl]pyridine-3-carboxamide
1-(5-methanesulfonamido-2-methylphenyl)-3-{1-oxaspiro[4.5]decan-3-yl}urea
(1S,5R)-6-benzyl-3-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3,5-dimethylphenyl)methyl]-4-(2-fluoro-4-methylbenzoyl)piperazin-2-one
1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
4-(ethylamino)-5-methyl-N-[3-(methylsulfanyl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-methyl-5-propyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
1-(2-methoxyphenyl)-4-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-yl)piperazine
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-(4-chloro-2-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)acetamide
N-ethyl-5-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}pyrimidin-2-amine
7-methyl-3-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-methoxy-N-{1-[1-(propane-1-sulfonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-(1H-imidazol-1-yl)-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
N3-[1-(4-fluorophenyl)ethyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(2,6-dimethylphenoxy)propyl]-N,3,5-trimethyl-1-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
1-[3-(azocan-1-yl)propanoyl]-N-(3-hydroxypropyl)piperidine-3-carboxamide
2-{4-[(3-ethylmorpholin-4-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
(2E)-3-(2-chlorophenyl)-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)prop-2-enamide
10-methoxy-5-(2-propyl-1,3-thiazole-4-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(4-fluorophenyl)-4-[3-(1H-imidazol-2-yl)benzoyl]piperazin-2-one
(1S,5R)-6-(4-chloro-3-methylbenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-ethoxy-5-{2-[(1-phenylethyl)amino]pyrimidin-4-yl}benzoic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
N-({4-[(dimethylamino)methyl]phenyl}methyl)-N-methyl-4-(piperidin-3-yl)benzamide
1-(carbamoylmethyl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]piperidine-3-carboxamide
N-[2-(4-hydroxyphenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
(2S,4S)-4-cyclopentaneamido-N-ethyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
2-(2,3-dimethoxy-5-methylphenyl)-N-methylpyridine-4-carboxamide
1-{2-[(5-methylhexan-2-yl)amino]ethyl}cyclopentan-1-ol
(1S,3R)-3-amino-N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)cyclopentane-1-carboxamide
(4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}phenyl)methanol
3-[(3R,4S)-1-[4-(ethylamino)pyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-cyclopentanecarbonyl-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-butyl-1-(2-methoxyphenyl)-4-(1-methylpiperidine-4-carbonyl)piperazin-2-one
1-(4-{[(4-methylphenyl)amino]methyl}benzoyl)piperidine-4-carboxylic acid
2,5,7-trimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide