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N-[2-(propylsulfanyl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-cyclopropyl-6-(4-methylphenyl)-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3R,5R)-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(3-methoxyphenyl)pyrrolidine
1-(2-{4-[(4-cyanophenyl)methyl]morpholin-3-yl}acetamido)cyclopentane-1-carboxamide
1-(1-benzylpyrrolidin-3-yl)-2-(1H-imidazol-4-yl)-1H-imidazole
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2,7,8-trimethylquinoline
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-(1H-pyrazol-4-yl)butan-1-one
4-hydroxy-N-[(2S)-1-methoxypropan-2-yl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
2-methyl-6-{2-[(pyridin-3-yl)amino]ethyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
4-[2-(3-methoxyphenoxy)ethyl]benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-yl]methanol
(1S,5R)-3-benzoyl-6-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-4-(trifluoromethyl)benzamide
3-{[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-methylbenzamide
4-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-imidazole-5-carboxamide
(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-(azocan-1-yl)-3-[4-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-{3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
4-(4-ethoxy-3-methylphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]butanamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
5-cyclobutyl-N-[1-(4-fluorophenyl)ethyl]-1,3,4-oxadiazol-2-amine
3-(1H-imidazol-2-yl)-6,8-dimethyl-1,2-dihydroquinolin-2-one
3-{[2-(dimethylsulfamoyl)ethyl]carbamoyl}-5-methoxybenzoic acid
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-methyl-2-{[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-(2-methoxy-5-phenylphenyl)-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]urea
4-methyl-2-(propan-2-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,3-thiazole-5-carboxamide
N-[(4-acetamidophenyl)methyl]-2-({[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}amino)acetamide
2-(3,4-dimethylphenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 3-(2-phenoxyethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
N-(3-methoxypropyl)-1-methyl-N-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-amine
1-methyl-9-(prop-2-en-1-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-{2-[1-(quinolin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
2-[4-(4-fluorophenyl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy]-1-(thiomorpholin-4-yl)ethan-1-one
2-[2-(dimethylamino)ethyl]-8-[2-(3-methoxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
6-cyclopentyl-2-methoxy-3-({[1-(propan-2-yl)piperidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1-methyl-2-phenylpiperazine
9-{[2-(methylsulfanyl)phenyl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-[(2-aminopyridin-3-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{5-[3-(4-fluorophenyl)propyl]-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
6-[(1-phenylethyl)amino]-1-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-N,N-dimethylpyrrolidin-3-amine
2-[(2-benzylbutyl)amino]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one