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1-[(4-methoxyphenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-2-(furan-2-yl)ethane-1,2-dione
2-amino-7-[3-(2-methylphenyl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
2-[(5-chlorothiophen-2-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
5-fluoro-2-[2-(2-phenylethyl)morpholine-4-carbonyl]-1H-indole
2-(2,3-dimethylphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
5-methyl-6-(morpholine-4-carbonyl)-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
1-{[5-(1-cyclopentylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
1-(2-chlorobenzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
[1-(2-chlorophenyl)-2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl]dimethylamine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(3S,4R)-1-(1,3-benzoxazol-2-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine-3-carbonitrile
N-(1-carbamoylcyclopentyl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-({1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({2-[4-(propan-2-yloxy)phenyl]ethyl})amine
7-(2-methoxyethyl)-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-4-[(5-{pyrazolo[1,5-a]pyridine-7-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]piperazine
methyl 3-(2-methyl-5-oxo-1,4-diazepane-1-carbonyl)benzoate
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-[(2-methylpyridin-3-yl)oxy]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-4-carboxamide
4-tert-butyl-6-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)-N-methylacetamide
3-[({4-benzyl-5-[1-(2-methylpropyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
5-[butyl(methyl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
1-[(prop-2-en-1-yloxy)carbonyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
5-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
9-[(5-chlorothiophen-2-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}azepan-3-amine
8-[3-(benzenesulfonyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,7S)-6-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(2,3-dihydro-1H-inden-2-yl)-4-{[1-(furan-2-ylmethyl)piperidin-4-yl]amino}pyrrolidin-2-one
N-(benzylsulfamoyl)-N-(2-methoxyethyl)-1-methylpiperidin-4-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(quinoxalin-2-ylmethyl)amine
5-cyclopropyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
9-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
3-ethyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1H-indole-2-carboxamide
1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1,3,3-trimethyl-6-[2-(4-methylpiperazin-1-yl)-6-(thiophen-2-yl)pyridine-3-carbonyl]-6-azabicyclo[3.2.1]octane
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
3-[1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)piperidin-3-yl]benzoic acid
N,N,9-trimethyl-3,9-diazaspiro[5.6]dodecane-3-sulfonamide
(1R,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-benzyl-3-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}benzamide
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)propanamide
2-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)benzonitrile