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N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-azaspiro[5.5]undecan-9-amine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
8-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-N-[(4-fluorophenyl)methyl]-4-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-3-(pyridin-3-yl)-N-(thiophen-3-ylmethyl)propanamide
(3S,9aR)-3-(cyclohexylmethyl)-8-(pyridin-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
(2S)-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-hydroxy-3-phenylpropan-1-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl]urea
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2-methyloxolan-2-yl)methyl]pyrimidin-2-amine
N-(1-{[2-(4-butyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}pyrrolidin-3-yl)-N-methylacetamide
4-methyl-6-[3-(2-phenylethyl)piperidin-1-yl]pyrimidin-2-amine
2-{4-[4-(pyridin-4-yl)piperazin-1-yl]quinazolin-2-yl}ethan-1-amine
N'-[2-(4-chlorophenyl)propyl]-N-cyclopentylbutanediamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyrrolidin-1-yl)acetic acid
11-[(3-ethoxypropyl)amino]-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-(dimethylamino)-2-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
N-methyl-N-[3-(oxolan-2-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N3-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-N1-(pyridin-3-yl)propane-1,3-diamine
4-(3,5-difluoropyridine-2-carbonyl)-1-(3,5-dimethylphenyl)piperazin-2-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
3-[(2R,3R,6R)-5-(1H-indole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
N-ethyl-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-(morpholin-4-yl)-3-[3-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
4-methyl-2-(pyridin-3-yl)-5-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrimidine
1-(2-methoxyphenyl)-4-{3-[methyl(1-methylpyrrolidin-3-yl)amino]propanoyl}piperazin-2-one
(2S,4R)-4-amino-N-ethyl-1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
N-({5-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-[4-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-(4-methylbenzoyl)-N-[1-(2-methylpropyl)piperidin-4-yl]piperidin-4-amine
1-{3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}ethan-1-one
1-{4-[(1,3-benzoxazol-2-ylmethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
N-[3-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)carbamoyl}amino)phenyl]-2-methoxyacetamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(2-methyl-1H-pyrrole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-methoxyphenyl)methyl]methylamine
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)thiophene-2-carboxamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-phenylpiperidine-1-carboxamide
3-(4-methylpyrimidin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
{1-[1-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-ol
1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(cyclohex-1-en-1-ylmethyl)-2-[(1-ethylpyrrolidin-2-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
2,7,8-trimethyl-N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]quinoline-4-carboxamide
2,5-dichloro-N-[(1-methylpiperidin-3-yl)methyl]benzene-1-sulfonamide
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2,2-dimethylpropan-1-one
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3-(2-methylphenyl)piperidine
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine