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N-benzyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
5-(2-fluorophenoxymethyl)-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-1H-pyrazole-3-carboxamide
5-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
1-[3-cyclopentyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-butyl-1,6-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
methyl 5-cyano-6-{3-[2-(dimethylcarbamoyl)ethyl]piperidin-1-yl}-2-methylpyridine-3-carboxylate
3-{[1-(4-methylpyrimidin-2-yl)pyrrolidin-3-yl]methyl}benzoic acid
1-[(1R,5S,6R)-6-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexan-3-yl]-2-methoxyethan-1-one
(1S,5R)-3-[2-(pyridin-3-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 2-{1-[3-(furan-2-yl)propanoyl]piperidin-2-yl}acetate
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6,7-dimethoxy-4-methylquinolin-2-amine
5-(azocan-1-yl)-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2-{2-[1-(benzenesulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-cyclobutyl-3-[(oxolan-3-yl)sulfamoyl]benzamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
(1R,7S)-6-(2,3-dihydro-1H-isoindole-2-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-methyl-4-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}benzene-1-sulfonamide
N-cyclopropyl-2-(1H-indazol-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
8-chloro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}quinoline-2-carboxamide
7-(cyclobutylmethyl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-3-(2-methylphenyl)-N-(oxan-4-yl)-3-phenylpropanamide
1-[3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenyl]ethan-1-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyrrolidin-1-yl)pyrrolidine
N-[(3R,4S)-4-cyclopropyl-1-(3-methylpyrazin-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
1-(3-chloro-2,6-dimethylphenyl)-3-(oxolan-3-yl)urea
2-methoxy-5-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)phenol
N-(pyridin-2-ylmethyl)-4-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N,5-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrazine-2-carboxamide
4-ethyl-3-(1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
(2R,4S)-4-hydroxy-1-(2-methyl-1,8-naphthyridine-3-carbonyl)piperidine-2-carboxylic acid
3-{3-[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]propoxy}pyridine
methyl 1-oxo-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,2-dihydroisoquinoline-7-carboxylate
N-[2-(4-sulfamoylphenyl)ethyl]spiro[2.5]octane-1-carboxamide
3-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-4H-chromen-4-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(4-chlorophenyl)methyl]-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-(cyclobutylsulfamoyl)-N-[2-(pyridin-4-yl)ethyl]benzamide
1-[(1-ethylpyrrolidin-2-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
1-ethyl-N,5-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-tert-butyl-3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(4-chlorophenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclobutane-1-carboxamide
2-(3-{1-[3-(morpholin-4-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-(2-phenoxyethyl)-1,4-diazepan-5-one