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2-amino-4-(4-chloro-1-methyl-1H-indazol-3-yl)-6-methyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
11-{[2-(4-chlorophenyl)ethyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-6-methylpyridine
2-[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]-N-(1,3-thiazol-2-yl)propanamide
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
4,4,4-trifluoro-3-({4-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)butanoic acid
methyl 1-[2-hydroxy-3-(4-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-[(3-hydroxypyrrolidin-3-yl)methyl]-6-methyl-2-(pyridin-3-yl)quinoline-4-carboxamide
ethyl 2-({3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenyl}amino)acetate
N-[3-(1H-pyrazol-5-yl)phenyl]-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
1-(5-fluoro-2-methylphenyl)-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}pyridine-3-carboxamide
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-4-methylpentane-1,2-dione
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-amino-6-methyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)pyrimidine-4-carboxamide
dimethyl(3-{2-[1-(pyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)quinoline-2-carboxamide
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
(4aR,8aS)-1-(oxane-4-carbonyl)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine
4-{4-[3-(3-fluorophenoxy)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
(4aS,7aR)-1-(4-methylpentanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
(4aR,7aS)-1-benzyl-4-[2-(methylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2,6-dimethoxy-4-methylphenyl)-N,N-dimethylpyridine-3-carboxamide
[(3R,4R)-1-(3,4-dimethylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(3S,4S)-4-cyclopropyl-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidine-3-carboxylic acid
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(5-methylfuran-2-yl)methyl]-2-phenylacetamide
2-(3-{[7-(1-hydroxy-2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(2,3-dimethylphenoxy)acetyl]-decahydro-1,6-naphthyridin-2-one
N-(3-hydroxypropyl)-1-(6-methyl-2-propylpyrimidin-4-yl)piperidine-3-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(pyrimidin-2-yl)pyrrolidin-3-yl]methanol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4,4,4-trifluorobutanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-acetamido-N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)benzamide
8-(1H-imidazol-4-ylmethyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]pyridine
2-(1H-indol-3-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
2,6-dimethyl-5-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
[(2S)-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
6-methyl-2-(2-{4-[1-(propan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
4-methyl-1-{2-[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3-triazole
6-oxo-N-[2-(pyridin-3-yloxy)propyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[2-(2-methoxyethoxy)phenyl]-3-phenylpiperazine-1-carboxamide