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2-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
6-[(oxolan-3-ylmethyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-[(cyclohexylamino)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}morpholin-2-yl)methanamine
1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-2-(1,3-thiazol-2-yl)piperidine
3-methyl-5-({4-[3-(prop-2-en-1-yloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1,2-oxazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(pyridin-2-yl)acetyl]pyrrolidine-3-carboxylic acid
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]-1-[4-(4-fluorophenyl)piperazin-1-yl]propan-1-one
N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-3-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3aS,6aR)-5-[6-(dimethylamino)pyrimidin-4-yl]-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1R,5S,8R)-3-[(5-ethylfuran-2-yl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
(1R,3s,6r,8S)-4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-ethyl-N-[(4-methoxyphenyl)methyl]acetamide
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1-(pyrimidin-2-yl)piperidine-4-carboxamide
N4-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
(3S,4R)-N-(4-chlorophenyl)-3-acetamido-4-(propan-2-yl)pyrrolidine-1-carboxamide
4-methoxy-N-(4-{4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]piperidin-1-yl}phenyl)benzamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-3-(5-methyl-1,2,4-oxadiazol-3-yl)benzamide
3-[2-fluoro-6-(propan-2-yloxy)phenyl]-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
2-(1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}piperidin-2-yl)ethan-1-ol
N-[2-(methylamino)ethyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[2-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
6-ethyl-N-[1-(2-methoxyphenyl)propan-2-yl]-N,1,5-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-[(diethylamino)methyl]-N-(4-methylpyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-(6-methoxynaphthalen-2-yl)-4-(5-methyl-1,3,4-oxadiazol-2-yl)morpholine
4-methylphenyl (7R,9aR)-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-cycloheptyl-2-{2-cyclopropyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl}-2-oxoacetamide
1-(3-methylbutyl)-2-oxo-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
[1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)piperidin-3-yl]methanol
2-(morpholin-3-yl)-1-(2-phenylpyrrolidin-1-yl)ethan-1-one
2-{2-[3-cyclopentyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
2-{[4-(1-phenyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(pyridin-4-yl)propan-1-one
[(3-ethoxy-4-methoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[(3R,4R)-3-hydroxy-1-(3-hydroxybenzoyl)piperidin-4-yl]pyridine-4-carboxamide
4-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2,1,3-benzoxadiazole
2-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(furan-3-carbonyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
4-[(2S)-1-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carbonyl]morpholine
1-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}piperidin-3-ol
6-[2-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-4-amine
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(1H-pyrazol-4-yl)butanoyl]piperidine-4-carboxylic acid