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1-(4-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]phenoxy}butyl)piperidine
5-(2-methylphenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,2,4-triazin-3-amine
4-[(2-fluorophenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carbonitrile
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-methyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N,N-dimethyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]azepan-4-amine
3-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]benzamide
N-cyclopropyl-N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-2-methylpropanamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
3-(cyclohexylmethyl)-5-(furan-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-3-carboxamide
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
1-(3,4,7-trimethyl-1H-indole-2-carbonyl)azetidine-2-carboxylic acid
4-methyl-3-{2-[2-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-4-(2-ethylpyrimidin-5-yl)-8-hydroxy-5H,6H-benzo[h]quinoline-3-carbonitrile
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-(1-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}[2-(diethylamino)ethyl]methylamine
(3R,4S)-1-(5-chloro-3-fluoropyridin-2-yl)-4-propylpyrrolidin-3-amine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
7-(1H-1,2,3-benzotriazole-5-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-[(3S,4R)-4-(propan-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-yl]methanesulfonamide
4-(5-acetylthiophene-2-carbonyl)-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
5-methyl-3-[2-(morpholin-4-yl)ethyl]-5-{1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-(cyclohexylmethyl)-2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]acetamide
1-methyl-2-[3-(2-methylphenoxy)azetidine-1-carbonyl]-5-phenyl-1H-pyrrole
4-{4-[(2,5-dimethoxyphenyl)methyl]piperazin-1-yl}-6-methoxypyrimidine
(3S,4R)-4-(3-methoxyphenyl)-1-(quinolin-5-ylmethyl)pyrrolidine-3-carboxylic acid
1-(2-ethoxyethyl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-ethyl-N-[3-hydroxy-1-(4-methylphenyl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,4R)-1-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
2-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}-1-(propan-2-yl)-1H-1,3-benzodiazole
methyl[(4-methyl-1,3-thiazol-2-yl)methyl]({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amine
3-[(dimethylamino)methyl]-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-3-ol
7-(cyclopropylmethyl)-2-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-(2-methoxyethyl)-3-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-amino-N-ethyl-1-[2-(pyridin-2-yl)acetyl]pyrrolidine-2-carboxamide
4-oxo-5-phenoxy-1-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxylic acid
1-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3-benzotriazole
N-(thiolan-3-yl)-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)(pentan-3-yl)amine
1-methyl-3-(propan-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
N-{[7-chloro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)furan-2-carboxamide
1-ethyl-4-({[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)pyrrolidin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-(oxolan-2-ylmethyl)acetamide
3-{1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one