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(3S,4S)-4-(morpholin-4-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-ol
N-[(2-fluorophenyl)methyl]-3-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}propanamide
1-(furan-2-carbonyl)-3-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}piperidine
4-chloro-1-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1H-pyrazole-5-carboxamide
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-methyl-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazine
3-[4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
1-{3-[(4,4-difluoropiperidin-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
ethyl 4-(4-{6-[ethyl(methyl)amino]pyrimidin-4-yl}piperazin-1-yl)piperidine-1-carboxylate
{2-[2-butyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]-2-oxoethyl}urea
2-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-N-(prop-2-en-1-yl)aniline
2-{[({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]methyl}-4-methoxyphenol
1-[2-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
6-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-(methylsulfanyl)benzamide
(2S,4S)-4-amino-1-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoic acid
5-(2-fluorophenyl)-4-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-2-(pyridin-3-yl)pyrimidine
ethyl 5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
4-(1-cyclobutanecarbonylpiperidin-3-yl)benzoic acid
N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]butanamide
N-ethyl-N-[2-(3-methylphenoxy)ethyl]-1-propyl-1H-pyrazole-5-carboxamide
N-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)acetamide
1-{4-[3-(2-methylphenoxy)azetidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
3-[2-(ethylsulfanyl)ethyl]-1-(4-fluoro-3-methoxyphenyl)urea
2-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
5-(3,4-dimethylphenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1,2-oxazole-3-carboxamide
2-[5-(3,4-dihydro-2H-1-benzopyran-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(3-methylpentan-3-yl)acetamide
1-ethyl-5-(2-methoxynaphthalen-1-yl)-1H,4H-pyrazolo[3,4-d]imidazole
(5-{4-phenyl-1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazol-5-yl}furan-2-yl)methanol
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
N-ethyl-N-methyl-2-{[1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
N-methyl-N-(2-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)methanesulfonamide
4-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]-3-methyl-1-phenyl-1H-pyrazol-5-amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-pyrazol-1-yl]acetamide
3-(3,5-dimethoxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
N'-[(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methyl]ethanediamide
methyl 5-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-[2-(3-fluorophenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-(methoxymethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-methoxy-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-4-carboxamide
2-methyl-5-[4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,7,8-trimethylquinoline-4-carboxamide
1'-(1-ethyl-1H-pyrazole-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cycloheptyl-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
(2S,4R)-N,N-diethyl-4-propanamido-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide