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N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-benzofuran-2-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
(2R,3R)-3-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-3-yl}-2-phenylethan-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methylacetamide
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1-(2-methoxyphenyl)piperazin-2-one
N-cyclopentyl-2-(methylamino)-N-[(3-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
(2R)-N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(5-fluoro-2-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-{[2-amino-6-(azepan-1-yl)pyrimidin-4-yl]amino}ethan-1-ol
2-(1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)ethan-1-amine
5-(1-benzoxepin-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N,3-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-(phenoxymethyl)furan-2-carboxamide
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)-3-(pyridin-4-yl)propanamide
2-(4-chlorophenoxy)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(1H-imidazol-4-ylmethyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
7-methoxy-4-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]quinazoline
N-{2-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]quinolin-6-yl}acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[3-(1H-indazol-1-yl)propyl]propanamide
2-benzyl-3-oxo-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazine-1-carboxamide
7-chloro-4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-(4,4-difluoropiperidine-1-carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
N-[1-(2-methanesulfonylethyl)piperidin-4-yl]imidazo[1,2-a]pyridine-6-carboxamide
5-[5-(butan-2-yl)-4-phenyl-1H-imidazol-1-yl]pentan-1-amine
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(1-methoxypropan-2-yl)piperidine
(3S,5S)-1-benzyl-N-[(4-chlorophenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
5-ethyl-2-{[4-(4-methyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
1-[(3-fluorophenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
4-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)-1-propylpyrrolidin-2-one
4-[2-amino-3-cyano-6-(trimethyl-1H-pyrazol-4-yl)pyridin-4-yl]benzoic acid
(3aR,6aR)-2-[2-(4-fluorophenoxy)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(furan-2-ylmethyl)(methyl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-(4-fluorophenyl)-N-methylmethanesulfonamide
1-(2,2-dimethylpropanoyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4-diazepane
N-{4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}acetamide
1-[(4aR,8aS)-1-[(2-hydroxynaphthalen-1-yl)methyl]-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
methyl 2-[methyl({3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}methyl)amino]acetate
N-(3-{4-ethoxy-3-[(methylamino)methyl]phenyl}phenyl)acetamide
4-[7-methoxy-6-(2-methoxyacetamido)-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl]-1H-pyrazole-3-carboxylic acid