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N-[2-(2-methoxyphenyl)ethyl]-5-phenyl-1,2,4-triazin-3-amine
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(2-methoxyethyl)piperidine
2-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
2-[(3-chlorophenyl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-(5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-methyl-3H-imidazo[4,5-b]pyridine
(1R,5S)-8-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octane
N-(2-hydroxypropyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-cyclopropyl-2-methyl-7-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyridine-3-carboxamide
1-{6-methyl-5-[5-(1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}-2-(methylsulfanyl)ethan-1-one
7-methyl-3-(3-phenyl-1,2-oxazole-5-carbonyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
8-(6-hydroxyhexyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1,9-dimethyl-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(3-chlorobenzoyl)-N-(3-chlorophenyl)piperidine-1-carboxamide
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}[(3-methylthiophen-2-yl)methyl]amine
7-(1,3-benzothiazol-2-yl)-4-(2-hydroxybenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)methanol
1'-(1-methyl-1H-indole-6-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
4-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-6-methylpyrimidin-2-amine
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-[(1S,5R)-3-[(3-cyanophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]pyrrolidin-3-ol
2-methyl-6-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-4-yl]pyrimidin-4-ol
2-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}benzoic acid
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-phenyl-1H-imidazol-5-yl)phenol
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
N-(oxan-2-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(4-{[(7-chloro-4-methylquinolin-2-yl)amino]methyl}oxan-4-yl)methanol
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-methyl-9-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-ethyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2,5-trimethyl-1H-pyrrole-3-carboxamide
3-(3-chlorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-hydroxyphenyl)-N-methylpropanamide
3-ethyl-6-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-ethyl-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethylpyrimidin-4-amine
2-[5-(3-cyclohexyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]acetamide
2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethan-1-ol
3-methyl-7-{[3-(naphthalen-2-yl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(quinolin-8-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(3,5-difluoro-4-methoxybenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(3,5-difluorophenyl)ethyl]-4-methyl-1H-imidazole-5-carboxamide
N-cyclopentyl-3-{[2-(thiophen-2-yl)ethyl]sulfamoyl}benzamide
1-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-1H-pyrazole-5-carboxamide
methyl 6-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carboxylate
N-(2,2-diphenylethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-(2,5-dimethylphenoxy)-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
(3R,4R)-4-(azepan-1-yl)-1-[1-(4-fluorophenyl)piperidin-4-yl]piperidin-3-ol