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1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}-4-phenylpiperazine
1-benzyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyrrolidine-2-carboxamide
1-[4-(ethylsulfanyl)phenyl]-3-(3-hydroxypropyl)-3-(1-phenylethyl)urea
6-hydroxy-N-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1,4-oxazepane-4-carboxamide
6-ethyl-4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyridin-2-one
3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}-7-methylquinolin-2-ol
1-methyl-2-oxo-8-(1,3-thiazol-5-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-benzyl-N-(3-hydroxy-2-methylpropyl)-1H-indole-2-carboxamide
4-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyrimidine
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]azepane
2-{4-[(2,6-difluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
(5-{1-[(8-methoxyquinolin-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
3-[(1-cycloheptylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-4-methoxybenzamide
N-(2-hydroxy-2-phenylethyl)-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-4-ylmethyl)propanamide
4-(4-chlorophenyl)-1-{5-methyl-4-[(oxolan-3-yl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperidin-4-ol
[1-cyclobutanecarbonyl-3-(3-methoxypropyl)piperidin-3-yl]methanol
N-[3-(morpholin-4-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
9-[(6-fluoroquinolin-2-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[2-(2,5-dimethoxyphenyl)-1H-imidazol-1-yl]-2-methyl-1H-1,3-benzodiazole
3-(4-fluorophenyl)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5-propyl-1,2-oxazole-3-carboxamide
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1-methyl-1H-indazol-3-amine
2-{2-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]pyrrolidin-1-yl}-4-methylquinazoline
9-(cyclopropylmethyl)-1-methyl-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(1s,4s)-4-aminocyclohexyl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(methylsulfanyl)propyl]-2-(5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}thiophen-2-yl)pyrrolidine
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylprop-2-en-1-yl)amine
9-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-3-oxa-9-azaspiro[5.5]undecane
(1S,5R)-3-(2-amino-6-methoxypyrimidin-4-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(2-methoxyphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-methoxypropyl)-N-(2-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{2-[4-(2-fluorobenzenesulfonyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
ethyl 2-(1-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazol-6-yl}-N-methylformamido)acetate
1-(3-ethylpiperazin-1-yl)-3-(pyridin-3-yl)propan-1-one
5-methyl-4-(4-methylpyrimidine-5-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
3-[1-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3-{[1-(quinoxaline-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-benzyl-4-cyano-N-(prop-2-en-1-yl)benzamide
6-methoxy-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
(2S,4S)-4-amino-N-methyl-1-{3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}pyrrolidine-2-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-methylpyridazin-3-amine
(2S)-2-{[4-(azocan-1-yl)-5-methylthieno[2,3-d]pyrimidin-6-yl]formamido}-4-methylpentanamide
N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[3-methyl-1-(pyridin-3-yl)butyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-5-methyl-1,3-oxazole-4-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-decahydro-2,7-naphthyridine-2-carboxamide