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1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-4-(thiophen-3-ylmethyl)piperazine
1-[4-(4-chloro-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidin-1-yl]ethan-1-one
2-({4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
5-methyl-5-[1-(4-phenylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
5-tert-butyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1,3,4-oxadiazol-2-amine
1-(2-methylfuran-3-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-ethyl-3-{[1-(5-methyl-1H-indazole-3-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(4-chloro-3-methylbenzoyl)pyrrolidin-3-yl]benzoic acid
4-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidine
2-(3-fluorophenyl)-4-(3,3,3-trifluoropropyl)pyrimidine
1-(2,6-dimethylpyridin-3-yl)-3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-methylfuran-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
1-[4-({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)piperazin-1-yl]ethan-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-(6-phenylpyridazin-3-yl)-decahydro-1,6-naphthyridin-2-one
2-(4-{[2-(cyclopentyloxy)phenyl]methyl}-1,4-diazepan-1-yl)-N,N-dimethylacetamide
(3S,4R)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(2-chloro-4-{[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}phenoxy)acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(diethylamino)acetamide
1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
3-{1-[1-(4-methoxyphenyl)-2,2-dimethylcyclopropanecarbonyl]azetidin-3-yl}pyridine
(2R,3S,6R)-5-(furan-2-ylmethyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1H-imidazole-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-(2,1,3-benzoxadiazol-4-yl)-N-benzyl-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(4-ethoxyphenyl)-2-propyl-1H-imidazole
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(2S,4R)-4-amino-1-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-N-methylpyrrolidine-2-carboxamide
2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-4-(trifluoromethyl)pyrimidine
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-4-yl]-2-phenylethan-1-ol
N-[1-(4-ethoxyphenyl)ethyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[methyl(2-phenylethyl)amino]-2-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
3-(4-hydroxyphenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-cyclopentyl-2-[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]butanamide
1-(3-fluoro-4-methylbenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
N-(cyclohexylmethyl)-2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]acetamide
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
cyclopentyl 4-(1,4-dioxane-2-amido)benzoate
8-(6,6-dimethyl-5-oxothiomorpholine-3-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-ethyl-6-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-{4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]morpholin-3-yl}acetamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
3,3-dimethyl-1-{4-[4-(1,3-oxazol-5-yl)phenyl]phenyl}urea
(1R,2S)-1-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2,3-dihydro-1H-inden-2-ol
1-[4-(oxan-2-ylmethoxy)phenyl]-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-cyclohexyl-N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
5-amino-N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide