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N-[(3R,4R)-3-hydroxy-1-(1H-indole-6-carbonyl)piperidin-4-yl]pyrazine-2-carboxamide
1-[(6-chloropyridin-3-yl)methyl]-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazine
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[2-(2-methoxyphenyl)ethyl]acetamide
5-[4-(thiomorpholine-4-sulfonyl)phenyl]pyrazin-2-amine
8-[(3-carboxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
9-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(butane-1-sulfonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
1-(4-methylpyridin-2-yl)-4-[4-(piperidin-3-ylmethyl)benzoyl]piperazine
N-butyl-N-ethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(2-benzyl-1,3-thiazole-4-carbonyl)piperidine-3-carboxylic acid
(3aS,6aS)-5-(6-methylpyridazin-3-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-1-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-4-ethylpiperidine-3,4-diol
1-(3-{[3-(3-ethylpiperazine-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
1-(cyclohexylmethyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-4-yl](pyridin-2-yl)methanol
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
[(5-chloro-2-methoxyphenyl)methyl][(1,3-dimethyl-1H-pyrazol-5-yl)methyl]ethylamine
2-amino-N-ethyl-6-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-4-carboxamide
8-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1-oxa-8-azaspiro[4.5]decane
1-(2-chlorophenyl)-4-(3-ethoxypropanoyl)-5-methylpiperazin-2-one
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-7-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
3-methoxy-1-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-N-(thiophen-2-ylmethyl)benzamide
2-(2-oxopyrrolidin-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
(1S,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-{5-[(2,3-dihydroxypropyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-1-phenylcyclohexane-1-carboxamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-[3-(aminomethyl)phenyl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
4-{1-[2-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}thiomorpholine
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-{3-[2-(3-cyanopiperidin-1-yl)-2-oxoethoxy]phenyl}propanamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(2-ethoxyphenyl)piperidine-1-carboxamide
(4aS,7aR)-1-(2-hydroxypyridine-3-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-4-oxo-1-(2-phenylethyl)-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
7-(2-hydroxyethyl)-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carboxamide
5-[(3-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1,2-oxazol-5-yl)methoxy]-2-methylpyridine
1-cyclopropyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
N-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine
2-{[(4-chloro-2-fluorophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(4aS,7aR)-1-[(2-ethoxyphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
6-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-[2-(butan-2-yloxy)-3-methoxyphenyl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide