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2-(2H-1,3-benzodioxol-5-yl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-[(6-chloropyridin-3-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
1-[2-(4-methylpentyl)morpholin-4-yl]-3-(pyridin-4-yl)propan-1-one
2-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
2-cyclopropyl-N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-(2-methoxyethyl)-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
1-(carbamoylmethyl)-N-{[5-(4-chlorophenyl)-1,2-oxazol-3-yl]methyl}piperidine-4-carboxamide
2-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-3-methyl-1H-indole
N-methyl-N-{2-phenyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
1-(3-chloro-4-fluorophenyl)-3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
4-{2-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylbenzene-1-sulfonamide
2-methyl-6-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
1,3-dimethyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(4-methanesulfonylmorpholin-2-yl)methyl]urea
{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
2-(1-ethylpiperidin-4-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]ethan-1-one
1-(1-methylpiperidin-4-yl)-4-(pyridazine-4-carbonyl)-1,4-diazepane-6-carboxylic acid
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrrolidine-2-carboxamide
4-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-6-(propan-2-yl)pyrimidin-2-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
9-[(3,4-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-6-(2-methylbutan-2-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
methyl 4-(5-{[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]propanoic acid
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
(1S,5R)-6-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidine
N-cyclopropyl-2,3-dimethoxy-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
5-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2,4-dimethyl-1,3-thiazole
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
3-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
ethyl 4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
N-(1-hydroxybutan-2-yl)-5-methyl-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide
2-(cyclopropylmethyl)-N-(oxan-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-methyl-1-(1-methylpiperidin-4-yl)-N-(propan-2-yl)piperidine-3-carboxamide
2-(1,7-dimethyl-1H-indole-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
7-(3-chlorophenyl)-4-cyclobutanecarbonyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine