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5-cyclobutanecarbonyl-1'-(piperidin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-ethylcyclohexane-1-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(3R,4S)-1-(1H-imidazol-4-ylmethyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
3-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
4-[(8-methoxyquinolin-2-yl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4,4-difluoropiperidine
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-one
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]quinoline
6-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4R)-3-ethyl-4-methyl-1-{pyrazolo[1,5-a]pyridine-2-carbonyl}piperidin-4-ol
(3S,9aR)-8-(naphthalene-2-carbonyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(2-hydroxy-7-methylquinolin-3-yl)-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
2-{2-[(3-oxopiperazin-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
9-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]naphthalene-1-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazin-2-one
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-5-phenyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
5'-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]
N-[4-methoxy-2-(2-methylpropanamido)phenyl]oxolane-2-carboxamide
{2-[4-(5-chloropyridine-2-carbonyl)morpholin-2-yl]ethyl}dimethylamine
(1S,5R)-N-(2-methylphenyl)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-N,N-dimethyl-2-oxo-decahydro-1,6-naphthyridine-6-sulfonamide
1-[1-(cyclopentylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-[1-(2-methylpropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-(2-ethoxypyridine-3-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
5-tert-butyl-4-({6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(1-benzyl-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
(3S,4S)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
1-[(4aR,8aS)-1-(2,2-dimethyloxane-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-cyclopropyl-5-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]pyrimidine
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
2-(dimethylamino)-N-[2-(furan-2-yl)ethyl]-2-(2-methylphenyl)acetamide
(3S,4R)-1-(1,1-dioxo-1λ6-thiane-4-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(4-methoxyphenyl)-5-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyrimidine
7-(2-hydroxyethyl)-2-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-(thiophen-2-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)butan-1-one
(3ar,6ar)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
{[5-(2,5-dihydro-1H-pyrrole-1-carbonyl)-2-ethylfuran-3-yl]methyl}diethylamine
4-(3-cyclohexylpyrrolidin-1-yl)-1-methylpiperidine