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1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
3-cyclopropyl-5-(5-methyl-1,3-oxazol-4-yl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-fluorobenzamide
2-(2-{[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
3-(2-methanesulfonamidoethyl)-1-[4-(4-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]urea
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-benzyl-3-ethyl-1-(6-methoxypyrimidin-4-yl)-1,4-diazepan-5-one
8-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-{6-methylimidazo[1,2-a]pyridin-2-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aR,7aS)-1-propanoyl-4-[(2,4,5-trimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[4-(1-methyl-1H-indole-6-carbonyl)piperazin-1-yl]-1,2-benzothiazole
N-{[8-(5-methylpyrimidin-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
3,3-diphenyl-N-[2-(1,3-thiazol-2-yl)ethyl]propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
4-ethyl-2-methyl-6-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-methyl-3-(2-methylpropyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4,4-difluoro-1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidine
4-(4-fluoro-2-methylbenzenesulfonyl)piperazine-2-carboxylic acid
3-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-[(4-carbamoylpiperazin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-methyl-4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-1,4,9-triazaspiro[5.5]undecane
2-(oxan-2-ylmethoxy)-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
2-(hydroxymethyl)-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-1,3-benzodiazole-5-carboxamide
2-[3-(5-methylfuran-2-yl)-5-(2-propyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-(3-fluorophenoxy)-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-benzothiazole
N-tert-butyl-1-cyclohexyl-5-[3-(diethylamino)pyrrolidine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-hydroxypyrazine-2-carboxamide
5-chloro-2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
1-[(5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}thiophen-2-yl)methyl]pyrrolidine
(3S,4S)-1-(3-methylbenzoyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2,2-dimethyloxane-4-carboxamide
7-(1-benzothiophen-3-yl)-4-[(2-ethylpyrimidin-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-2-{[2-(5-methyl-1H-pyrazol-1-yl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-cyclopropyl-4-(3-fluoro-2,4-dimethylphenyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N,N-diethyl-1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
5-[4-(benzyloxy)piperidine-1-carbonyl]-1-ethylpiperidin-2-one
1-(3-methoxyphenyl)-3-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)urea
(4aR,7aS)-1-methyl-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(prop-2-en-1-yl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carboxamide
methyl 6-{1-methyl-2,6-dioxo-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinolin-8-yl}pyridine-2-carboxylate
2,3-dimethyl-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide
N4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
7-methoxy-3-[(3-phenylpiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one