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1-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pentane-1,2-dione
(3aR,6aR)-2-(2-hydroxyethyl)-5-[1-(2-phenylethyl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2Z)-3-(3-fluorophenyl)-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
N,2-dimethyl-3-(2-oxo-5,5-diphenylpiperidin-1-yl)propanamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-amino-2-(2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethyl)pyrimidin-4-ol
2-(3,5-difluorophenyl)-N-(1,4-dioxan-2-ylmethyl)acetamide
1-(2-{4-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidin-2-amine
(2S)-3-methyl-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}butanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-[(dimethylamino)methyl]-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-ol
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[1-(pyrimidin-4-yl)ethyl]piperidin-4-amine
N-butyl-6-oxo-1-(prop-2-en-1-yl)-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
2-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
4-chloro-2-(2-ethoxypyridin-3-yl)phenol
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-7-methoxy-N-methyl-N-(2-methylpropyl)quinoline-4-carboxamide
3-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5-methyl-6-(4-methylphenyl)pyridine-3-carbonitrile
2-[(4aR,7aS)-4-[(4-fluoro-2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
(2R,3R)-3-(2-methyl-1H-imidazol-1-yl)-1'-(1H-pyrazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-methoxy-1-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-indole-2-carboxamide
1-(butan-2-yl)-3-methyl-5-(2,3,4-trimethoxy-6-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
6-[2-(methoxymethyl)piperidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(2R,3R)-1'-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
2-(2-oxo-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-2-azaspiro[4.6]undecan-3-one
(4-{[4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
1-{[1-(hydroxymethyl)cyclopentyl]methyl}-1-methyl-3-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]butanamide
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-(1H-indol-3-yl)-1H-1,2,4-triazol-1-yl}acetic acid
3-butanamido-N-(cyclopropylmethyl)-N-propylbenzamide
4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-{3-[(2-methoxyphenyl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-1-methyl-1,2-dihydropyridin-2-one
1-cyclopentyl-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1,4-diazepane
1-{2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)morpholin-2-yl]ethyl}-3-ethylurea
(3R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3,4,4-trimethylpyrrolidin-3-ol
13-(5-ethylfuran-2-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
4-(2-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)morpholine
4-{4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl}pyrimidine-5-carboxylic acid
1-{2-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide