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(1S,5R)-6-benzyl-3-(2-methoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2-chlorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]furan-2-carboxamide
(1R,7S)-N-methyl-4-oxo-3-(pentan-3-yl)-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}propanamide
4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
ethyl 4-(6-{[5-(methoxymethyl)furan-2-yl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
1-[(3-methoxyphenyl)methyl]-3-phenyl-6-(pyrazine-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1H-indol-2-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-{4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}quinoline-4-carboxylic acid
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-methyl-2-(3-methylphenoxy)butan-1-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-cyclopentylethan-1-one
1-[2-(2-hydroxyethyl)phenyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
2-cyclopropyl-8-(8-methoxyquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1-cyclohexylpiperidin-3-yl)-4-(4-methoxyphenyl)piperazine
1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-({[(3-{2-[4-(2-cyclopentylacetyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-methylphenoxymethyl)piperidine
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-hydroxypropan-1-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentane-1,2-dione
4-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
3-methyl-3-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-(5-pentyl-1,3,4-thiadiazol-2-yl)urea
3-{imidazo[1,2-a]pyridin-2-yl}-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
2-hydroxy-N-({1-[1-(2-methylphenyl)piperidin-4-yl]piperidin-3-yl}methyl)acetamide
2-[4-(3-acetylphenyl)phenyl]-N-methylacetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
3-[4-(2-amino-1,3-thiazol-4-yl)phenyl]-N-cyclopropylbenzamide
7-{[3-(4-methoxyphenoxy)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazole
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(pyridine-3-carbonyl)-1,4-diazepane
1-[(4-methylphenyl)methyl]-4-[4-(4-methylpyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
8-methyl-5-{4-[1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}quinoline
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylic acid
1-(2-ethyl-6-methylphenyl)-5-oxo-N-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-({1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
1-benzoyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
(1S,5R)-3-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl][2-methyl-2-(piperidin-1-yl)propyl]amine
1-[(4-chloro-3-fluorophenyl)methyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
8-(1-benzofuran-2-ylmethyl)-3-benzyl-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1H-imidazole
1,3-dimethyl-2,6-dioxo-N-[2-(propane-2-sulfonyl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(2,3-dimethylquinoxaline-6-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
5-chloro-3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
5-methyl-N-[3-(morpholin-4-yl)propyl]-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
4-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-[1-(2,3-difluoro-4-methoxybenzoyl)piperidin-3-yl]-2-phenylethan-1-one
N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide