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4-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}thiomorpholine
2-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}furan-3-carboxamide
1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-[5-(methanesulfonylmethyl)pyridin-2-yl]-2-methoxyquinoline
3-chloro-N-(2-methoxyethyl)-4-({1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}propan-1-one
2-{4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]morpholin-3-yl}-1-(pyrrolidin-1-yl)ethan-1-one
3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-(4-fluorophenyl)-1H-1,2,4-triazole
1-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(thiophen-2-yl)propan-1-one
4-(2-ethylphenyl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-(5-chlorothiophene-2-sulfonamido)-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
1-{[1-(3-chloro-4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-3,3-dimethylurea
2-(dimethyl-1,2-oxazol-4-yl)-1-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)ethan-1-one
3-chloro-2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
1,3-dimethyl-N-(pentan-3-yl)-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
6-methyl-5-(pyrimidin-5-yl)-1,3-benzothiazol-2-amine
2-(1-{[3-(2-methylphenyl)phenyl]methyl}pyrrolidin-2-yl)ethan-1-ol
3-[5-(7-methyl-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
4-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
1-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(thiophen-2-ylmethyl)piperazine
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](3-phenylprop-2-yn-1-yl)propylamine
5-(2,3-difluorophenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-hydroxyacetamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
2-amino-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyridine-4-carboxamide
8-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-ethyl-1-methyl-3-({1-[(2,3,4-trifluorophenyl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
N-(2-fluorophenyl)-3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
N-[4-(4-methoxyphenyl)phenyl]-4-methyl-1,4-diazepane-1-carboxamide
1-(3-chloro-2,6-dimethylphenyl)-3-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
3-(2-chlorophenyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
1-[(2-fluorophenyl)methyl]-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]piperidin-2-one
6-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[4-(2-aminoethyl)phenyl]methyl}-3-[(dimethylamino)methyl]piperidin-3-ol
2-[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]-1-methyl-1H-1,3-benzodiazole
2-{5-[3-(1H-imidazol-1-yl)propyl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}pyridine
(1R,5R)-N,N-dimethyl-6-(3-phenoxypropyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-6-methoxyphenol
(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methanamine
3-({8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decan-1-yl}methyl)pyridin-2-amine
(3R,4R)-4-ethyl-1-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]piperidine-3,4-diol
N-(4-chloro-2-fluorophenyl)-2-({1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}amino)acetamide
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
1-(2-ethoxyethyl)-N,3-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-methylpyrimidine