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(3aR,6aR)-2-cyclopentyl-5-[(4-hydroxy-3-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4S)-4-cyclopropyl-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
3-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]quinoline
N-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
1-methyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-methoxy-2-(2-methoxypyrimidin-5-yl)quinoline
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-chloro-5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidine-3-carbonyl}pyridine
1-[1-(2,6-diaminopyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidine-1-carbonyl)piperazine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxan-4-amine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclohex-3-ene-1-carboxamide
2-{4-[(tert-butylcarbamoyl)amino]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
N-[(3-methoxyphenyl)methyl]-3-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}propanamide
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[2-(morpholin-4-yl)propyl]amine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[ethyl(methyl)amino]pyridine-3-carboxamide
N4-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-6-(propan-2-yl)pyrimidine-2,4-diamine
2-amino-4-[2-(ethylsulfanyl)pyrimidin-5-yl]-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-(1H-pyrazol-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
1-methyl-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}azepane
4-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2-(3,4-dichlorophenyl)morpholine
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]cyclopropane-1-carboxamide
9-[(2R,3S)-2-amino-3-hydroxybutanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
2-methoxy-N-{3-[1-(methoxymethyl)cyclobutaneamido]phenyl}benzamide
N-(2,3-dimethylquinoxalin-6-yl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
2-(2-propyl-1H-1,3-benzodiazol-1-yl)-N-(2,2,2-trifluoroethyl)propanamide
2-(dimethylamino)-N-[1-(hydroxymethyl)cyclopentyl]-2-(4-methylphenyl)acetamide
1-[(2S)-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-1-yl]ethan-1-one
1-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-ethylacetamide
1-{[1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
(4aS,8aR)-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(2S)-2-cyclohexyl-2-[(6-cyclopropylpyrimidin-4-yl)amino]ethan-1-ol
3-cyclopropyl-4-(8-methoxy-2H-chromen-3-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-(4-tert-butyl-1,3-thiazol-2-yl)acetamide
4-[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]benzoic acid
3-[(3R,4S)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
4-methyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-[(3aR,6aR)-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(pyridin-3-yl)piperazine
2-methyl-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]-1H-imidazole
5-(1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-N,N-dimethylthiophene-2-carboxamide
6-chloro-3,4-dimethyl-7-[1-(3-methyl-1H-1,2,4-triazol-5-yl)ethoxy]-2H-chromen-2-one
(3S,4S)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
5-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine