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{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
(4aS,8aR)-1-(2-methylpropyl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-decahydro-1,6-naphthyridin-2-one
1-(3-cyclopropyl-5-{[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)isoquinoline
5-(1-{3-[(3-fluorophenyl)carbamoyl]propanoyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-{[3-(methylsulfanyl)propyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
2-{3-[2-(trifluoromethoxy)phenyl]phenoxy}acetamide
(4aS,7aR)-1-(3-methylbutanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
11-(cycloheptylamino)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-[(dimethylamino)methyl]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]furan-2-carboxamide
4-[(6-methylpyridin-3-yl)oxy]-1-[2-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
N-cyclopropyl-4-[(6-acetamidoquinolin-2-yl)methyl]piperazine-2-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(4-hydroxyphenyl)ethyl]benzamide
2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-benzyl-1-(5-ethylpyrimidin-2-yl)piperidin-4-ol
1-[(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
8-({3-[(2-chlorophenyl)methoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
N-{3-[(pyridin-3-yl)amino]propyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3R,5S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
4-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,4S)-1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
5-(2-chloro-4-fluorophenoxymethyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(4-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenyl)acetamide
N,N-dimethyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
5-(2,6-difluorophenoxymethyl)-N-(1H-indol-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}pyrimidine
6-methyl-2-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
N-(1-benzothiophen-5-ylmethyl)-1,1-dioxo-1λ6-thiane-4-carboxamide
2-[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-2-yl]pyridine
4-[2-(3-methoxyphenoxy)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxylate
6,8-dimethyl-2-[({1-oxa-8-azaspiro[4.5]decan-3-yl}amino)methyl]quinolin-4-ol
(2Z)-2-fluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-phenylprop-2-enamide
7-(4-fluoro-2-methylbenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[(3-methylquinoxalin-2-yl)methyl]cyclopropanamine
N-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
5-(1-{2-[(4-chlorophenyl)methoxy]ethyl}-1H-1,2,3-triazol-4-yl)pyrimidine
6-(2-aminoethyl)-N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyrimidin-4-amine
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1-propanoylpiperidine-3-carboxamide
5-fluoro-1-methyl-2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-[2-(ethylsulfanyl)phenyl]-2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
3-cyclohexyl-N-(1H-indol-6-ylmethyl)-1H-pyrazole-4-carboxamide
1-{3-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]ethan-1-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(5-{[4-(2-methylphenyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
3-methyl-4-{2-methyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-1-(2-methylpropyl)piperazin-2-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperazine
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-[1-(cyclohexylmethyl)piperidin-3-yl]propanamide