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1-{[(3R,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
(3R,4S)-1-(4-aminopyrimidin-2-yl)-3,4-dimethylpiperidin-4-ol
(2R,6S)-4-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
1-(3-hydroxypropyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
(4aR,7aS)-1-{2-[4-(hydroxymethyl)-4-methylpiperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({7-[(4-acetamidophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[2-(dimethylamino)propanoyl]piperidine-4-carboxylic acid
(1S,5R)-6-(5-fluoropentyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-[(methylsulfanyl)methyl]-2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridine
5-(pyridin-3-ylmethyl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-[(1R,5R)-6-{[3-(trifluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-({3-methyl-7-[2-(thiophen-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
1-(2-{[2-(methylsulfanyl)pyrimidin-4-yl]amino}ethyl)pyrrolidin-2-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1,3-trimethyl-1H-pyrazole-4-carboxamide
2-amino-6-[4-(piperidin-1-yl)phenyl]-4-(piperidin-3-yl)pyridine-3-carbonitrile
[2-ethoxy-5-({3-[(4-fluorophenyl)amino]piperidin-1-yl}methyl)phenyl]methanol
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(quinolin-4-yl)-1,4-diazepan-5-one
(1-methyl-5-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
(3S,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}benzamide
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-[4-(1H-pyrazol-5-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
ethyl 4-benzyl-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidine-4-carboxylate
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(pyridin-2-ylsulfanyl)ethan-1-one
4-methyl-5-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]-1,3-thiazole
4-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine-1-carboxamide
2-[2-(dimethylamino)pyrimidin-5-yl]-N-(1-methylpiperidin-3-yl)quinoline-4-carboxamide
4-methyl-2-(4-methylpiperazin-1-yl)-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrimidine
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-2-(1H-pyrazol-3-yl)pyridine
ethyl 1-(1-acetylpiperidine-4-carbonyl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
2-{4-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]morpholin-3-yl}acetic acid
2-(4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)-1-methylazepane
2-(2-acetylphenyl)pyridine-3-carbonitrile
3-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-6-methylphenol
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
2-(2-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
7-(2-hydroxypropanoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(2,5-difluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)urea
[(1-benzylpiperidin-4-yl)methyl][(2-ethylpyrimidin-4-yl)methyl]methylamine
1-cycloheptyl-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S,9aR)-8-(4-fluorobenzoyl)-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-benzyl-5-oxopyrrolidin-2-yl)propanamide
1-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
3-amino-1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidine-3-carboxylic acid
9-(2-hydroxybenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[(3-methylpyridin-4-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one