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N-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
7-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-{4-[2-(pyrrolidin-1-yl)acetyl]morpholin-3-yl}acetamide
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
5-(3-benzoylpiperidine-1-carbonyl)-N-ethyl-4-methyl-1,3-thiazol-2-amine
2-(adamantan-1-ylsulfanyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
3-(3-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}-1H-indol-1-yl)propanamide
1-[2-(cyclohexylsulfanyl)ethyl]-3-[4-(morpholin-4-ylmethyl)phenyl]urea
N-[2-(dimethylsulfamoyl)ethyl]-2-(1,3-thiazol-4-yl)acetamide
ethyl 1-{2-[(furan-2-ylmethyl)carbamoyl]ethyl}piperidine-2-carboxylate
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
(5-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}furan-2-yl)methanol
1-{4-[2-(3-aminoazepan-1-yl)-2-oxoethyl]phenyl}imidazolidin-2-one
N,N-dimethyl-3-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)benzamide
13-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
2-[methyl({4-methyl-5-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-[(4-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-pyrazole
3-(3-{5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propyl)pyridine
1-({[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
4-ethyl-5-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-3-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)propanamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidin-2-amine
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
1-{6-[2-(trifluoromethyl)morpholin-4-yl]pyridin-3-yl}ethan-1-one
2-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
3-[(3R,4S)-1-[(3,4-difluorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-(4-fluorophenyl)-N-[(1-methylpiperidin-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-4-(trifluoromethyl)benzamide
[(3R,4S)-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-ethyl-2-(4-hydroxy-3-methylphenyl)pyridine-4-carboxamide
(3S,4R)-1-[2-(azepan-1-yl)acetyl]-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
4-cyclobutanecarbonyl-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-4-(pyrimidin-2-yl)piperazine-1-carboxamide
1-(2-{[1-(4-oxo-3,4-dihydroquinazolin-3-yl)propan-2-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
3-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}-1,3-oxazolidin-2-one
(3S,4S)-4-[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]-1-(propan-2-yl)pyrrolidin-3-ol
4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-1-(propan-2-yl)pyrrolidin-2-one
(2S,4R)-4-hydroxy-N-[4-methoxy-2-(2-methylpropanamido)phenyl]pyrrolidine-2-carboxamide
N-[4-(2-chloro-6-methoxyphenyl)-2-ethylphenyl]acetamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)(quinolin-4-ylmethyl)amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-[2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-(oxolan-2-ylmethyl)-5-propyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
4-(5-chloro-2-methoxyphenyl)-5-(propan-2-yl)pyrimidine
4-(4-chlorophenoxy)-1-(furan-3-carbonyl)piperidine
(4aR,7aS)-1-[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N,N-dimethylfuran-2-carboxamide