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2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]azepan-2-one
2-{3-[3-(3-methylphenyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
5-[4-(aminomethyl)piperidin-1-yl]-2-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
6-(3-chlorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(pyrrolidine-1-sulfonyl)ethyl]amine
2-amino-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
1-(5-methyl-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine
1-butyl-3-(oxan-4-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
4-[4-(dimethylamino)benzoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-(cyclohexylmethyl)-3-hydroxy-3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}piperidin-2-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-4-methyl-1H-imidazole-2-carboxamide
4-(3,5-dimethylbenzoyl)-1-phenylpiperazin-2-one
1-cyclohexyl-4-(6-cyclopropylpyrimidin-4-yl)-1,4-diazepane
8-[(6-chloro-2H-chromen-3-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
4-[(2-fluorophenyl)methyl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,4-diazepan-5-one
N,1,5-trimethyl-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-3-carboxamide
N,N-dimethyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-chloro-4,6-dimethyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(furan-2-yl)-N-[1-(pyridin-3-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide
3-(4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
1-[(8-methylquinolin-5-yl)methyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
2-(2-amino-6-methylpyrimidin-4-yl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(thiophen-3-ylmethyl)piperidin-4-yl]methanesulfonamide
N-[(3R,4R)-1-[(2-fluoro-4-methoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-[(4-fluorophenyl)methyl]-1-{2-[(3-methylthiophen-2-yl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-(1H-imidazol-2-ylmethyl)-3-(3-methoxyphenoxymethyl)piperidine
4-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-2-methylphenol
(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-7-{[(2-fluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-cyclopropanecarbonyl-N-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-amine
3-[4-(2-methylphenoxy)piperidin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
1-{3-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}-1H-pyrazole
1-(3-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
8-(1-hydroxypropan-2-yl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4,4,4-trifluoro-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
5-({[1-(3-methoxyphenyl)propan-2-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(2-methylpropyl)-2-(2-oxopyrrolidin-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
3-cyclopropyl-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-1H-pyrazole-5-carboxamide
5-butyl-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
2-(4-fluorophenyl)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-2-(piperidin-1-yl)acetamide
5-(3,3-diphenylpropanoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-oxoethyl]azonan-2-one
2-[(6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)amino]ethan-1-ol
7-(8-hydroxy-5,7-dimethylquinoline-2-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N,8-dimethyl-3-{[methyl(oxan-2-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one