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(3R,4R)-1-(6-chloro-2H-chromene-3-carbonyl)-3-cyclobutyl-4-methylpyrrolidin-3-ol
N-[(3R,4R)-3-hydroxy-1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
1-(2-ethoxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
9-(2-methoxyethyl)-1-methyl-4-(oxan-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
N-[3-(3-cyanopyrazin-2-yl)phenyl]acetamide
8-[(4-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(4-methoxyphenyl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N5-(1-benzylpiperidin-4-yl)-1-cyclopentyl-N3,N3-diethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{[5-(1-cyclopropanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
N,4,6-trimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-(2-ethylpyrimidine-5-carbonyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
4-(1H-1,3-benzodiazol-1-yl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine-4-carboxylic acid
3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
1-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]piperidin-4-ol
N-(4-acetylphenyl)-3-cyanopiperidine-1-carboxamide
4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
[(3R,4S)-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}propanamide
1-{4-[2-(4-methylpentyl)morpholin-4-yl]piperidin-1-yl}ethan-1-one
4-[(2R)-2-hydroxy-2-(naphthalen-2-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)pyridine-3-carbonitrile
4-{2,2-dimethyl-3-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]propyl}morpholine
8-[2-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrrol-1-yl)pyridine
N-[2-(ethanesulfonyl)ethyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
(3R,4R)-4-cyclobutyl-3-methyl-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-4-ol
2-methoxy-3-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
5-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(pyridin-3-yl)pyrimidine
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-6-fluoro-3,4-dihydroquinazolin-4-one
(3R)-3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-[2-methyl-5-(propan-2-yl)pyrimidin-4-yl]benzamide
4-[1-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1H-imidazol-2-yl]benzoic acid
(4aS,7aR)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1,2-oxazol-3-ylmethyl)-3-[(pyridin-2-ylmethyl)sulfamoyl]benzamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[2-(propylamino)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
(2-{1-[2-(difluoromethoxy)benzoyl]piperidin-2-yl}ethyl)dimethylamine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(pyridin-3-yl)acetamide
ethyl 1-[(4-chlorophenyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
7-(1,3-benzothiazol-2-yl)-4-[2-(oxolan-3-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,6-dimethyl-4-{[4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]methyl}phenyl acetate
3-{5-[(2-oxo-1,2-dihydropyrimidin-1-yl)methyl]-3-phenyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-{2-[4-(benzyloxy)-4-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)spiro[2.3]hexane-1-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-[(1-methylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
8-(2-amino-2-methylpropyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-chloro-4-[2-(pyrrolidin-3-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine