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8-(4-chloro-3-methylphenyl)-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]ethan-1-one
4-methyl-3-[(2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}acetamido)methyl]benzoic acid
1-{6-hydroxy-4-[(3-methylpyridin-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
1-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]cyclopropan-1-amine
4-{7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane-3-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
2-(5-acetylthiophen-3-yl)-N-methyl-N-(oxan-2-ylmethyl)acetamide
2-[(4-ethylcyclohexyl)formamido]-N-[(1-methylpiperidin-3-yl)methyl]acetamide
2-(3-{[3-(2-methylpropyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
8-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,4-difluorophenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
2-propyl-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
3-[5-(6-methoxypyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2,6-dihydroxy-N-methylbenzamide
1-(2-methoxy-5-methylphenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
3-(3-fluorophenyl)-4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperazin-2-one
2-(dimethylamino)-8-(8-methylquinolin-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(1-propylcyclopropyl)carbamoyl]pyrrolidine-2-carboxylic acid
N-ethyl-2-(3,4,5-trifluorophenyl)pyrimidin-4-amine
2-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
5-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,5R)-3-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4-diazepane
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]butan-1-one
1-(oxolan-3-ylmethyl)-4-(pyrimidin-2-yl)-1,4-diazepane
6-chloro-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-2-carboxamide
1-cyclohexyl-N-[(5-methoxy-1H-indol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-phenyl-3-(4H-1,2,4-triazol-4-yl)propan-2-ol
6-(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-2-methylpyrimidin-4-ol
{4-[({3-azaspiro[5.5]undecan-9-yl}amino)methyl]oxan-4-yl}methanol
9-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1,3-benzothiazol-2-ylmethyl)-3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-(1-{7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-3,5-dimethyl-1-phenyl-1H-pyrazole-4-sulfonamide
2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}propane-1,3-diol
2-(1H-pyrazol-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
N-(isoquinolin-5-ylmethyl)-N-methyl-3-(2-oxoazepan-1-yl)propanamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(5-ethyl-2-methylpyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2-aminoethyl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
3-[4-(1-cyclopropanecarbonylpiperidine-4-carbonyl)piperazin-1-yl]-2,5-dimethylpyrazine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylfuran-3-carboxamide
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-(quinolin-5-ylmethyl)acetamide
2-(2-fluorophenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
2-methanesulfonamido-N-{1-[(4-methylphenyl)methyl]cyclopropyl}propanamide
(2S,4R)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-4-hydroxypyrrolidine-2-carboxamide
2-methyl-4-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)-6-(1H-pyrazol-1-yl)pyrimidine
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-5-phenylpyridin-2-amine