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(2R)-2-amino-N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-4-methylpentanamide
1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-ethyl-8-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(propan-2-yl)-2-(4-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperazin-1-yl)acetamide
(3aS,6aR)-5-(5-propylthiophene-3-carbonyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-ethylpyrimidin-2-amine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methoxy-2-methylbenzamide
7-(cyclopropylmethyl)-2-[3-(2-oxoazepan-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine-2-carboxylic acid
1-(2-methyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
2-[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[(2-methylphenyl)methyl]acetamide
4-[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(3,5-dimethoxyphenyl)-3-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]propanamide
1-(4-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-(2-aminoethyl)-N-[2-(dimethylamino)butyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
N-[1-(4-methylphenyl)cyclopropyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-methyl-9-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[(2-methoxyphenyl)methyl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
4-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-1-(1H-indazol-5-yl)piperazin-2-one
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-(methanesulfonylmethyl)piperidine
2-[(4-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}phenyl)(methyl)amino]ethan-1-ol
4-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}benzoic acid
2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]ethan-1-ol
(3S,7S)-5-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)propanamide
N-phenyl-5-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrimidin-2-amine
5-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
(1R,5R)-6-[(2-chloro-6-fluorophenyl)methyl]-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
N-(4-{1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
methyl 5-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-5-oxopentanoate
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
1-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-ol
(2S,4R)-4-(furan-3-amido)-N-methyl-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)propanamide
7-(cyclohexylmethyl)-2-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}acetamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[4-(furan-2-yl)phenyl]piperidin-4-amine
1-{2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
3-[(2R,3R,6R)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(4aS,7aR)-1-(5-chlorothiophene-2-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3,6,7-trimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N,N-dimethyl-4-({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)butanamide
1-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2,3-dihydro-1H-inden-2-yl}piperidine