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1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(2-phenoxyphenyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4S)-4-amino-5-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-5-oxopentanoic acid
(3S,4S)-4-cyclopropyl-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
2-phenyl-5-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
3-[(4aR,7aS)-4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5-{1-[(5-chloro-2-hydroxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
(2S)-2-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)propanamide
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
benzyl N-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}pyrrolidin-3-yl)carbamate
5-{1-[2-(1,2-benzoxazol-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
(1R,5S,8S)-3-[(3,5-dimethoxyphenyl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-{[1-(5-ethoxyfuran-2-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methyl-1-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-ethyl-3-(piperidin-4-ylmethyl)-1-[(3,4,5-trifluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,6R)-4-[2-methyl-2-(morpholin-4-yl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[3-(2-methoxyethyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(3S,4S)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
4-{1-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]cyclohexyl}morpholine
(2S,4S)-4-(3,5-difluorobenzamido)-N-(1H-imidazol-2-ylmethyl)-1-methylpyrrolidine-2-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-[1'-(2-ethylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
methyl 7-oxo-9-(3-phenylpropoxy)-3-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(1-methylcyclopropyl)benzamide
(1S,5R)-3-cyclohexanecarbonyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-methyl-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(2-amino-3-cyano-6-cyclobutylpyridin-4-yl)-2-chlorophenoxy]acetamide
(2S,4R)-4-amino-N-ethyl-1-(4-methoxy-3-methylbenzenesulfonyl)pyrrolidine-2-carboxamide
(4aS,8aR)-6-(4-methyl-1,3-thiazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[3-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-3-oxopropyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-3-(1H-pyrazol-4-yl)benzamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-methyl-7-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(1,2-oxazol-5-ylmethyl)benzene-1-sulfonamide
(2R)-1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(methoxymethyl)pyrrolidine
N-(5-chloro-2-methoxyphenyl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
4-methoxy-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
3-ethyl-N-(furan-3-ylmethyl)-N,5-dimethyl-1,2-oxazole-4-carboxamide
1-benzyl-5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(2-acetamidoacetyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-{2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl}-4-(propan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-oxo-2-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidin-1-yl]ethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2-(2-methoxyethyl)morpholine
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2-ethylphenoxy)azetidin-1-yl]propan-1-one