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3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]pyridazine
N-(pyrrolidin-3-yl)-3-{[3-(1H-1,2,3-triazol-1-yl)propyl]sulfamoyl}benzamide
6-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-N-ethylpyridine-3-carboxamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)pent-4-enamide
2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]-1-(thiomorpholin-4-yl)ethan-1-one
4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}morpholine
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-phenyl-1,2-oxazole-3-carboxamide
3-(hydroxymethyl)-1-{[3-(pyridin-2-yl)phenyl]methyl}piperidin-3-ol
methyl 3-{[(1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
N-[1-(cyclohexylmethyl)piperidin-3-yl]-4-(1H-pyrazol-4-yl)butanamide
N-methyl-1-phenyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
methyl 5-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)-2-hydroxybenzoate
2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-N-(1-methyl-1H-pyrazol-3-yl)acetamide
1-({2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}methyl)cyclohexan-1-ol
1-(2-chlorophenyl)-2-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
4-[(1-{1-azabicyclo[2.2.2]octan-3-yl}piperidin-4-yl)oxy]-3-chloro-N-cyclopentylbenzamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-benzyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-{4-[1-(3-chloro-2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
4-[1-(2-ethoxyethyl)piperidin-3-yl]-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2,3,4-trifluorobenzoyl)pyrrolidin-3-yl]methanol
ethyl (4aS,8aR)-6-(3-chloro-2-fluorobenzoyl)-decahydro-1,6-naphthyridine-4a-carboxylate
5-(methoxymethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(3,5-difluorophenyl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
5-[4-(dimethylsulfamoyl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N'-({1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}methyl)ethanediamide
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N-dimethylpyrimidin-4-amine
2-[2-benzyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]acetamide
2-methoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}pyrimidine-5-carboxamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[(2-methoxyphenyl)methyl]piperidine-3-carboxamide
3-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(pyridin-3-yl)acetamide
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
1-{[3-(2-methylphenyl)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(piperidin-4-yl)acetamide
1-[2-(2-ethoxypyridin-3-yl)pyridine-4-carbonyl]-4-methylpiperazine
4-ethyl-5-methyl-2-[3-(pyridin-4-yl)azetidin-1-yl]pyrimidine
2-methyl-3-{[3-(pyridin-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole
4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazine-1-carboxamide
2-amino-6-(2-amino-5-methyl-1,3-thiazol-4-yl)-4-[2-(propylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
4-benzyl-3-ethyl-1-(2-hydroxyacetyl)-1,4-diazepan-5-one
N-methyl-N-(2-phenylethyl)-5-[(3-propoxypiperidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide