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7-(2-cyclohexylethyl)-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenol
(3R,4R)-1-(2-methanesulfonylethyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(2S)-2-{[(2,5-dimethylthiophen-3-yl)methyl]amino}propanamide
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-phenylazepane
N-[(3R,4S)-4-cyclopropyl-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
(1R,3S)-7-(3-fluoropyridin-2-yl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
3-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}piperidin-3-ol
N-cyclopropyl-2-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
9-(8-hydroxyquinolin-2-yl)-1-methyl-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(2-methoxyphenyl)ethyl]benzamide
N-butyl-3-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(2-fluoro-4-methoxyphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
2-(3-fluorophenoxymethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1,3-oxazole-4-carboxamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)(quinoxalin-2-ylmethyl)amine
N-butyl-N-[(2E)-3-phenylprop-2-en-1-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
1-{2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
8-[2-(azocan-1-yl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-{methyl[2-(methylamino)ethyl]amino}pyridine-3-carboxamide
5-(2-{2-[(2-amino-9H-purin-6-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-(1-methoxybutan-2-yl)-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-cyclopropyl-9-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[1-(6-ethylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
8-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
(3aR,6aR)-2-[2-(3-chlorophenyl)acetyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-amino-4-(furan-2-yl)-5-methyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)piperidin-2-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-methyl-5-[1-(oxolan-3-yl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(carbamoylmethyl)acetamide
6-({3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N2,N2-dimethyl-N4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
1-{4-[(2-cyclopentylethyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-(3-methyl-1H-pyrazol-4-yl)-3-(pyrrolidin-1-yl)pyrazine
ethyl 1-(2H-1,3-benzodioxol-4-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-[(2R,3R,6R)-5-(2-aminopyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3,6-trimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
2-(3-fluorophenoxymethyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-[methyl({4-methyl-5-[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-[(2-chlorophenyl)methyl]-4-(pyrazin-2-yl)morpholine
methyl 4-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-5-methylthieno[2,3-d]pyrimidine-6-carboxylate