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N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-5-(propan-2-yl)thiophene-3-carboxamide
[(2S,6S)-11-methoxy-4-(4,4,4-trifluorobutyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
[1-(6-methoxypyrimidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-(3-ethylphenoxy)-N-(2-methyl-1,3-benzothiazol-5-yl)azetidine-1-carboxamide
(3-{2-[1-(4-fluoro-3-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-[2-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenoxy]propanamide
N-methyl-5-(phenoxymethyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propane-1,2-diol
2-(dimethylamino)-7-(9H-fluorene-9-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(2-{1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
2-amino-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-6-(propan-2-yl)pyrimidine-4-carboxamide
4-[2-amino-3-cyano-6-(2,5-dimethylfuran-3-yl)pyridin-4-yl]benzamide
N4-[3-(1H-imidazol-2-yl)propyl]-5,6-dimethylpyrimidine-2,4-diamine
3-(2,3-dihydro-1H-inden-5-yl)-1-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}urea
1-[(2,3-dichloro-4-methylphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
1-[3-(3-fluorophenyl)benzoyl]-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-cyclohexyl-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-methyl-3-(naphthalen-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-ethyl-1H-pyrazol-5-yl)-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-fluoro-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-5-sulfamoylbenzamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
[(5-ethylfuran-2-yl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
2-amino-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}quinazoline-6-carboxylic acid
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2-(2-phenylethyl)piperidine
N-[1-(4-methanesulfonylphenyl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(3-hydroxyphenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
N-[2-(4-methoxyphenyl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
2-[3-(2-methylpropyl)-5-[(2S)-1-methylpyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl]pyridine
4-{2-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{[6-(6-methylquinolin-3-yl)pyrimidin-4-yl]amino}ethan-1-ol
5-[2-(methylsulfanyl)ethyl]-4-phenyl-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)prop-2-ene-1-sulfonamide
(3S,4R)-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(1-{1-[(2,3-difluoro-4-methoxyphenyl)methyl]piperidin-4-yl}ethyl)dimethylamine
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidine-4-carbonitrile
5-chloro-N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-sulfonamide
methyl (1S,3S,3aR,6aS)-3-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-5-ethyl-1-(hydroxymethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[1-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]methanesulfonamide
N-[3-(1H-imidazol-5-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
1-[(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
4-(methoxymethyl)-6-[4-(1H-pyrazol-1-yl)phenyl]pyrimidine
3-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
N-[(2R,4R,6S)-2-cyclohexyl-6-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]oxan-4-yl]acetamide
N-[2-(1-benzylpiperidin-4-yl)ethyl]morpholine-2-carboxamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide