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1-[2-hydroxy-5-(2-methoxypyridin-3-yl)phenyl]ethan-1-one
5-ethyl-2-[(E)-2-phenylethenyl]pyrimidine
3-cyclopentaneamido-N,4-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-methanesulfonyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepane
N-cyclopropyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
3,5-dimethyl-4-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenol
8-methyl-2-propyl-N-(pyridin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(cyclopropylmethyl)-2-(1-methyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridazine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-[3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
(2R,6S)-1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
1-methyl-3-(propan-2-yl)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
{1-[(5-chlorothiophen-2-yl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
[(4-fluorophenyl)methyl][(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](pyridin-4-ylmethyl)amine
ethyl 1-(1H-indol-3-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[3-(2-methoxyethyl)-5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1H-1,2,4-triazol-1-yl]benzoic acid
2-chloro-N-cyclohexyl-5-(1H-pyrazol-1-yl)benzamide
4-[(3-fluoro-4-methoxyphenyl)methyl]-2-[(4-methoxyphenyl)methyl]morpholine
3-(1-ethyl-1H-pyrazol-4-yl)-2,4,5-triazatetracyclo[11.4.0.02,6.07,12]heptadeca-1(17),3,5,7,9,11,13,15-octaene
(1S,5R)-6-[(5-fluoro-2-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-6-[3-(benzylsulfanyl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(dimethylcarbamoyl)amino]-N-[2-(5-methylthiophen-2-yl)ethyl]acetamide
6-phenyl-2-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3,4,5-tetrahydropyridazin-3-one
3-amino-1-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
1-ethyl-3-(piperidine-1-carbonyl)-N-[3-(pyridin-4-yl)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2,3-dimethyl-5-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzene-1-sulfonamide
(3S,4S)-1-(2-methylpyrimidine-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-(1-ethyl-5-oxopyrrolidin-3-yl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(4-{[2-(naphthalen-2-yl)ethyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]-N,N-diethylpyrrolidin-3-amine
ethyl 4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1H-pyrazole-3-carboxylate
3-{[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
N-cyclohexyl-3-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylformamido)propanamide
2-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-2,3-dihydro-1,2-benzothiazol-3-one
2-(ethylsulfanyl)-5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)pyrimidine
1-(3,4-dichlorophenyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazine
1-methyl-4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazine-2-carboxylic acid
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(3-methyl-1,2-oxazol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
8-(5-acetyl-4-methylpyrimidin-2-yl)-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(dimethylamino)ethyl]-N-methyl-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
ethyl 4-(3-phenylpropyl)-1-(thian-4-yl)piperidine-4-carboxylate
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
2-(3,4-dichlorophenyl)-4-(4-methylpyrimidin-2-yl)morpholine
2-{[(1-ethyl-1H-indol-6-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
N-{[3-(cyclopentyloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-2-(thiophen-3-yl)acetamide