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1-ethyl-4-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
4-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
6-methyl-2-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-cyclopropyl-2-(methylamino)-N-{[4-(methylsulfanyl)phenyl]methyl}pyridine-3-carboxamide
N-[2-(oxan-2-yl)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
(1R,5S,8R)-8-(dimethylamino)-N-{4-[(trifluoromethyl)sulfanyl]phenyl}-3-azabicyclo[3.2.1]octane-3-carboxamide
N,2,6-trimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}quinoline-3-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxamide
(1S,2S)-2-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}cyclohexan-1-ol
3-(1H-1,3-benzodiazol-2-yl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
4-[1-(trimethylpyrimidin-4-yl)piperidin-4-yl]morpholine
N-methyl-3-{methyl[(2-methyl-1,3-oxazol-4-yl)methyl]amino}butanamide
3-(2,4-difluorophenyl)-1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
N-methyl-N-(oxolan-3-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-({5-[(3-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}morpholine
3,5-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2-oxazole-4-carboxamide
3-(2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,3-diazinane-2,4-dione
N-(2,3-dimethylphenyl)-3-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropanamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrrol-1-yl)ethan-1-one
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-5-(propan-2-yl)-1,3-oxazole
4-[(2S)-2,6-diaminohexanoyl]-1-phenylpiperazin-2-one
2-(3-methoxyphenoxymethyl)-N-[(4-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
2-{ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}-N-(4-methylphenyl)propanamide
1,3,7-trimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1H-indole-2-carboxamide
N-tert-butyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-{[3-(methylsulfanyl)propyl]amino}benzene-1-sulfonamide
2-(dimethylamino)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(4-methylphenyl)ethan-1-one
methyl N-{2-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}carbamate
2-(5-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-[(3S,4R)-1-(5-fluoropyrimidin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
4-chloro-3-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-1-methyl-1H-indazole
methyl[1-(4-methylpyridin-2-yl)propan-2-yl](2-phenylethyl)amine
8-(isoquinolin-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(2S)-2-amino-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1H-indol-3-yl)propanamide
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
(4R)-N,3-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1,3-thiazolidine-4-carboxamide
N-[1-(3-phenylpropyl)piperidin-3-yl]-4-(thiophen-2-yl)butanamide
3-(1H-1,3-benzodiazole-5-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-{3-[4-({[1-(morpholin-4-yl)cycloheptyl]methyl}amino)piperidin-1-yl]phenyl}cyclopropanecarboxamide
1-[4-(1H-pyrazol-3-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
5-(2-chlorophenyl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]furan-2-carboxamide
(butan-2-yl)[(4-methanesulfonylphenyl)methyl](pyridin-4-ylmethyl)amine
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(3-methoxybenzoyl)piperazine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3-methoxypyrazin-2-yl)piperazin-2-one
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(4-fluorophenyl)ethyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-(3-phenylpyrrolidin-1-yl)acetamide