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N-[4-(3-methoxyphenyl)phenyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
2-[(4-chlorophenyl)sulfanyl]-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-ethyl-N-(4-hydroxybutan-2-yl)acetamide
3-[(4-cyclopentylpiperazin-1-yl)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
1-(4-fluorophenyl)-3-{[1-(2-methylpropyl)piperidin-3-yl]methyl}urea
2-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-{3-[(2,6-dimethylphenyl)carbamoyl]phenyl}-5-methylpyrazine-2-carboxamide
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
9-[(3R)-3-hydroxy-3-phenylpropyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-cycloheptyl-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidin-2-one
5-(5-fluoro-2-methoxyphenyl)-2-(propan-2-yl)-1,3-thiazole
(2S,4S,5R)-1,2-dimethyl-4-{[(5-methyl-1H-pyrazol-3-yl)methyl]carbamoyl}-5-phenylpyrrolidine-2-carboxylic acid
N1-(2,5-difluorophenyl)-N3-ethylpyrrolidine-1,3-dicarboxamide
(5S)-5-({[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
N-ethyl-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-3-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-oxo-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1,3-oxazolidine-4-carboxamide
3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-(propan-2-yl)propanamide
ethyl 4-(2-phenoxyethyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-4-carboxylate
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(4-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methanol
2-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}pyridine
5-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-[(3-carbamoyl-1,2,4-oxadiazol-5-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(2,4-dimethoxyphenyl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
6-ethyl-3-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1,5-dimethyl-1,2-dihydropyridin-2-one
(2R)-2-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
3-(pyridin-3-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
4-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}pyrimidin-2-amine
N-ethyl-2-(4-ethylpiperazin-1-yl)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)acetamide
5-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
1-(1-methyl-1H-pyrazole-4-carbonyl)-2-(2-phenylethyl)piperidine
4-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-propyl-1,3,4-oxadiazol-2-amine
2-(1-benzothiophen-7-yl)-4,6-dimethylpyridine-3-carboxamide
4-(4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
2-(2,3-dimethylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
2-(2,4-dichlorophenoxy)-N-[1-(1H-imidazol-1-yl)butan-2-yl]acetamide
5-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3,7-dimethyl-11-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecane
(1R,5S,6S)-N-methyl-3-[(2-methylpyrimidin-5-yl)methyl]-N-(1H-pyrazol-5-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
8-(2,3-dimethyl-1H-indole-7-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(4-fluorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-oxobutanamide
1-[1'-(2-methyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[3-(hydroxymethyl)quinolin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol