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4-chloro-1-methyl-3-{[(1S,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1H-indazole
1-[(3-methoxyphenyl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-phenyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1H-1,2,3,4-tetrazole
1-[2-(4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperazine
2-(2-methoxyethyl)-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-hydroxyphenoxy)ethan-1-one
3-(5-{[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-({1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(5-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
1-(2-{5-[(2,5-dimethylphenyl)methyl]-1,2,4-oxadiazol-3-yl}ethyl)pyrrolidin-2-one
1-(2-hydroxy-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
4-{4-[(3-ethenylphenyl)methyl]piperazin-1-yl}pyrimidin-2-amine
1-[cyclohexyl(methyl)amino]-3-{2-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}propan-2-ol
4-{3-[4-(2-hydroxyethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
1-(2-fluorophenyl)-4-[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
N-ethyl-N-[(1R,2R)-2-hydroxycyclohexyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(3S)-3-amino-3-{[(3-methylphenyl)methyl](propan-2-yl)carbamoyl}propanoic acid
N-(cyclohexylmethyl)-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-3-ol
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[2-(pyridin-3-yloxy)propyl]acetamide
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-N-(thiophen-3-yl)piperidine-1-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
7-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidine-1-carbonyl]-1,3-diazepane-2,4-dione
(2R,3R,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(pyridin-2-yl)propanamide
1-{[4-(2-methylpropyl)phenyl]methyl}-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(pyrrolidine-1-carbonyl)-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazine
2-(azepane-1-sulfonyl)-2,7-diazaspiro[4.5]decane
2-(1,3-benzothiazol-2-ylmethyl)-4-[4-(4-cyclohexylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-oxo-1,2-dihydroquinazoline-4-carboxamide
3-[1-benzyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
N3-(1-benzothiophen-2-ylmethyl)-N5-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(dimethylamino)-1-phenylethyl]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{[3-(3-methylphenyl)-1H-pyrazol-4-yl]formamido}-N-phenylpropanamide
2-{4-[(4-fluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
methyl (2R,4S)-4-hydroxy-1-(2-methoxypyridine-4-carbonyl)piperidine-2-carboxylate
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamido]acetic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-ethyl-1H-pyrazole-4-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(2R,3R)-1'-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{4-[(3-methoxyphenyl)methyl]-1-(naphthalene-2-sulfonyl)piperidin-4-yl}methanol
N-(butan-2-yl)-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(thiophen-3-ylmethyl)propanamide
4-{[(1R)-2-hydroxy-1-phenylethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid